ImpiloAmalungiselelo

Medicine "Trimetazidine". izinkomba

"Trimetazidine" - umuthi okhuthaza ukuzinza lokugayeka kokudla kumaseli wadalula ischemia noma hypoxia. Kusho cishe ngokuphelele futhi kuqhathaniswa matasa ngokushesha. I bioavailability zomuthi - 90%. Ubuningi kwakwakhe esebenzayo egazini ifinyelela isiqongo ngemuva kwamahora amabili. imikhiqizo Reaction excreted ngokusebenzisa izinso umchamo.

mshini wezenzo

Umuthi kuvimbela nokwehlisa izinga intracellular ATP, inikeza umsebenzi evamile iziteshi ulwelwesi ion. Umuthi futhi inikeza transmembrane ezokuthutha sodium ne-potassium ion nokugcina homeostasis. Kusho "Trimetazidine" okubonisa ukuthi isicelo okuzokwenza inikezwe ngezansi, kubamba namachibi of okunamafutha acid. Lokhu kuqinisekisa isivikelo ischemia. Ukushintsha ama namachibi glucose ne acid okunamafutha kubangela imithi antianginal. Phakathi ukulinga izilwane, kwatholakala ukuthi lesi sidakamizwa lisiza ekulondolozeni kwezitho zomzimba neurosensory futhi inhliziyo namandla umzimba ngezikhathi ischemic ka exacerbations. Ngenxa umsebenzi zomuthi incipha ngobungako lactic intracellular kanye nezinga izinguquko yokucucuza transmembrane ion. Ngaphezu kwalokho, izidakamizwa kunciphisa kokuziphatha futhi yokufuduka polynuclear neutrophil e reperfusion ischemic kanye nezicubu kwenhliziyo, kunciphisa ubukhulu umonakalo esivimba amanzi. Ngesikhathi esifanayo it is hhayi waphawula nemiphumela yayo hemodynamics.

Medicine "Trimetazidine": Ubufakazi

Umuthi Kufanele umise uchwepheshe. Kunconywe ukuba self-medicate. Ngaphansi akukho udokotela pathologies angabeka "Trimetazidine"? Izinkomba ukusetshenziswa kwezimali ngendlela elandelayo: cochle-vestibular iziyaluyalu imvelo ischemic (inzululwane, ukulahlekelwa kukuzwa, tinnitus), iziyaluyalu semithambo ezifana ischemic ingxenye chorioretinal. Umuthi nayo iqondiswa iziguli nokuvimbela ukuhlaselwa angina (njengoba monotherapy noma ukwelashwa).

I umthamo lwemithi

Lapho ukwabela izindlela "Trimetazidine" (izinkomba ukusetshenziswa zichazwe isihloko) is kunakwe kusho ukubekezelelana, kobukhulu isifo. Njengoba ojwayelekile, ukuphuza imithi ngaso 40-60 mg ngosuku. ethola imvamisa - 3.2 p / d.

Izimo, imiphumela emibi izidakamizwa "Trimetazidine". nobufakazi

Umuthi akunconyelwe iziguli abakhulelwe noma lactating, hypersensitive ukuba izingxenye. Izibuyekezo iziguli ukuthatha izidakamizwa, ngokuvamile, omuhle. Ngokusho iziguli, lesi sidakamizwa "Trimetazidine" izinkomba ukusetshenziswa okuye ezichazwe ngenhla, legciwane eliphansi imiphumela emibi. inkinga Common ukusabela nomzimba. Njengomthetho, kwenzeka ngenxa hypersensitivity. Ochwepheshe batusa ukuthi ukubukeka ukulunywa, ukuqubuka, isikhumba ukusabela kabi komzimba kanye nezinye imiphumela emibi ngenkathi ngokuthatha izidakamizwa ukubona udokotela. Kunconywe ukuba ashintshe isilinganiso semithi oyidlayo ku izimali zabo.

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