Impilo, Amalungiselelo
"Sedalia": yokusetshenziswa, Izimo, ukubuyekezwa
Yini sedatives kanye nemithi yokunciphisa ukucindezeleka zaziwa kuwe? Ethandwa kakhulu phakathi kodokotela abathengi ujabulele imithi kwemizwelo isimame ezifana "Sedalia". Izibuyekezo futhi imfundo zomuthi ethulwa ngezansi. Futhi e mathiriyeli lo sihloko ukubaluleka wakwambula, ukufundwa kanye anezakhi ezikhethekile.
Packaging izidakamizwa, ukubunjwa yayo, umumo
"Sedalia" - amaphilisi we-lenticular wangakwesokunxele, camera futhi ibekwe endaweni contoured aluminium ucwecwe iphakethe. Izithako main zomuthi yilezi: lithium carbonate, amazambane isitashi, talc, i-calcium stearate, povidone, hypromellose, polysorbate, tropeolin futhi titanium dioxide.
izidakamizwa
Kuyini isimame isimo ezifana "Sedalia"? Iziyalezo yokusetshenziswa Lithi normalizes isimo sengqondo kanye akakubangeli ukucobeka jikelele. Futhi, lolu izidakamizwa has antimanic, sine futhi isenzo antidepressant.
Ukuphumelela kwezidakamizwa kokucubungula lithium-ion, sodium ion kukhona abantu abamelene nani. Ngokusho imiyalelo, bona azixoshe kubo kusukela amaseli bese ukunciphisa umsebenzi bio kagesi-izinzwa ubuchopho.
Kufanele kuqashelwe ukuthi le isithako zomuthi kunomthelela nokwahlukana esasizosheshisa of ama biogenic. Ngakho, lo lokuhlushwa serotonin futhi norepinephrine emisipheni ubuchopho kuyehla, futhi ukuzwela izinzwa of hippocampus nezinye izindawo yesenzo sakhe ukukhuphuka Dopamine.
Lokhu ejenti baxhumana lipids, okuyinto akhiwa ngesikhathi umzimba inositol. Ngezinye ngemithamo zokwelapha, ke amabhlogo umsebenzi owodwa inositol-phosphatase futhi kunciphisa lokuhlushwa inositol neuronal ehilelekile ukulawulwa ukuzwela neuronal.
Umphumela ozuzisayo lithium e migraine kungenxa izamba histamine obuhlukahlukene futhi serotonin e-platelet. Futhi izakhiwo zalo antidepressant kubangelwa sithuthukiswe serotonergic umsebenzi bese wehlise ukulawulwa receptor beta-adrenergic.
izinkomba pharmacokinetic
Uma uthatha le imithi emva kokudla, it is matasa kusukela amathumbu kanye ifinyelela isiqongo salo e-plasma ngemva cishe 9 amahora. Leli thuluzi asisho abophe ukuze amaphrotheni, kodwa lingena isithiyo esinomhlapho futhi excreted e ngobisi lwebele.
Umuthi akuyona akheka futhi excreted ngu izinso e imali 95% (ngo emathunjini - ngaphansi kuka-1%, bese nge - mayelana 4-5%).
Izidakamizwa "Sedalia": Ubufakazi
Kwezinye izimo, bebheka bonke izidakamizwa kungenziwa Kunconywa yokwamukelwa? Ngokuvamile, lokhu kusho okunqunywe ngoba ukwenama sengqondo isigaba ekuvimbeleni exacerbations ka sengqondo (isimo) odabuka ezahlukene, ulaka (kuhlanganise ukuluthwa utshwala ezingamahlalakhona), ngeziphambeko ngokobulili, psychopathy futhi sezidakamizwa. Ngaphezu kwalokho, izidakamizwa esebenzayo ngokuvamile sisetshenziswa UMeniere Syndrome, ukuluthwa izidakamizwa psychotropic kanye migraine.
Uvala ukusetshenziswa kwezidakamizwa
Lapho hhayi ukusebenzisa amaphilisi sine "Sedalia"? Yokusetshenziswa ibika ukuthi lokhu imithi contraindicated uma hypersensitivity kuya izithako zako, ukuhlinzwa okukhulu, wegazi, futhi ibele futhi esikhathini ukukhulelwa.
Ngokucophelela okukhulu imithi kwemizwelo isimame ezinqunyiwe izifo zenhliziyo, isimiso sezinzwa esiyinhloko, psoriasis, isifo sikashukela, i-hyperthyroidism, hyperparathyroidism, futhi ukwehluleka kwezinso.
Tablets "Sedalia": yokusetshenziswa
Njengoba izindlela okuxoxwe okufanele zisetshenziswe? It is ezithathwe umlomo emva kokudla. Kulokhu, lo umthamo wansuku zonke sehlukaniswe kane. amaphilisi Kugcine kumele kwenziwe kusihlwa, noma kunalokho, ngaphambi kokulala.
Ngokuvamile, umthamo kokuqala nsuku zonke nomuthi kuyinto 0.6-0.9 r ne ukwenyuka kancane ku-1.2 g Ngemva kwalokho, inani lakhuphuka lafika ku-izidakamizwa 0.3 g futhi kushintshwe 1.5-2.1 g usuku ngalunye
Ungalokothi idlule umthamo wansuku zonke imithi, okungukuthi ukusetshenziswa ezingaphezu kuka 2.4
Isikhathi ukwelashwa imithamo ngenhla 2 g singemaviki lange 1-2. Uma nomuthi isetshenziselwa prophylactic, ke monotherapy ezigulini ingatholakala ekugcineni njalo igazi lokuhlushwa lithium ezingeni 0.4-0.8 mmol / l (izinyanga ezingaphezu kwezine ngalokho eziyisithupha).
Uma izimpawu of sengqondo ukwenama ukunqampunwa, umthamo wansuku zonke zomuthi kuyehla iviki elilodwa ngaphambi prophylactic (isb ukuba 0.6-1.2 g).
Lapho izimpawu nokuboniswa inani izidakamizwa kwandile futhi.
isinyathelo uhlangothi
izidakamizwa Antidepressant "Sedalia" kungabangela imiphumela engasi mihle ezifana:
- ukuba buthakathaka kwezicubu, inhliziyo isigqi neziyaluyalu, isandla eliqhaqhazelayo;
- hyperreflexia, ubuthakathaka, ukuqunjelwa, ukozela;
- ukuhambisana iziyaluyalu (administration ezingamahlalakhona), ukoma owandiswayo;
- ukungasebenzi yegilo indlala, leukocytosis;
- hemodyscrasia, kukhuphuke isisindo emzimbeni.
amacala ukweqisa izidakamizwa
Ngesikhathi ukusetshenziswa ebulilini zomuthi ngokuthi "Sedalia", intengo oboniswe ngezansi, isiguli bangezwa Isakhiwo sazamazama, ukuba buthakathaka kwezicubu, dysarthria, amajaqamba ezinzima, ukuhlanza, ukudideka, nesiyezi, ukungakuthandi ukudla, isifo sohudo, angaboni kahle, ukozela, isicanucanu futhi polyuria. Kulokhu, ukumisa izidakamizwa kanye nokwelapha lingaze.
ukuxhumana
Ngingakujabulela yini neminye imithi "Sedalia" ithebhulethi? Yokusetshenziswa ngokuvumelana ekusebenzisaneni ezilandelayo:
- Lapho ukuphatha ngesikhathi esisodwa ACE inhibitor, "Indapamide", futhi ama-NSAID isisu (thiazide) kungadala imiphumela ezinobuthi futhi nokwenyuka lokuhlushwa lithium egazini.
- Lapho kuhambisana ukusetshenziswa amalungiselelo iodine kwandisa ingozi ukwephulwa indlala yegilo.
- reception Parallel ne-sodium ne-hydrogen carbonate xanthine nemikhiqizo ithuthukisa inqubo ekususeni lithium kanye umchamo, okuyinto kunciphisa kakhulu ukuphumelela izidakamizwa.
- With ukusetshenziswa ngesikhathi esisodwa izidakamizwa incipha nge phenothiazines ukumuncwa yayo kusukela pheshana emathunjini, kanye lokuhlushwa yayo egazini. Lokhu kwandisa lokuhlushwa lithium ngaphakathi amaseli kanye izinga yayo excretion ne umchamo.
izincomo ezithile
iziguli ephelile, iziguli esezikhulile kuyadingeka ukuze ulungise lwemithi nokushintsha kokudla nokufakwa.
Ezinsukwini ezingu-30 zokuqala zokwelashwa kufanele ukulawula lokuhlushwa lithium egazini njalo ngesonto.
Phakathi ukwelashwa ayikwazi ukuphuza utshwala.
izidakamizwa Okufanayo futhi izindleko
Izidakamizwa "Sedalia" -, sine ngempumelelo kakhulu futhi fast-esebenza. Njengomthetho, intengo uyahluka ruble 120-150. Zuza izidakamizwa ezinjalo kungaba yisiphi izidakamizwa. Uma lokhu kusho ukuthini kuwe ayitholakali, kungase kuthathelwe indawo ontanga ezifana "Lithium carbonate", "UMikhali", "Litosan-SR", "Kvilonum", "Kontemnol".
Ngenxa yokuthi lezi zimali anezici ezabo isicelo, angasetshenziswa kuphela izincomo kadokotela.
Izibuyekezo
Yini imiyalezo ingatholakala kwi izidakamizwa "Sedalia"? Izibuyekezo iziguli nodokotela izokwethulwa manje.
Ezinye iziguli bathi kuyinto sine iphumelela kakhulu futhi ayibizi kakhulu. Abanye abasebenzisi bahlale bekhononda ngezinto iqiniso lokuthi lokhu izidakamizwa inemiphumela eminingi engemihle. Njengomthetho, ngemuva kokuthola iziguli anda isisindo futhi ibonakala zingavuvukalanga. Ngaphezu kwalokho, ngokuvamile lo izidakamizwa antidepressant kubangela abantu bengasinaki, ukucobeka jikelele, Ukoma okukhulu, ukozela, futhi arrhythmia.
Ngokuphathelene amazwana wezazi, bona ukubika ukuthi lapho kahle akhethiwe ngomthamo, kanye nokuqapha njalo wegazi lithium leli thuluzi ngempumelelo.
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