ImpiloAmalungiselelo

Yikuphi-analog "riboksin" ukukhetha: amathiphu kanye nokubuyekeza

izidakamizwa steroid - iqembu izidakamizwa, lo mshini eyinhloko esenzweni okuhloswe ngalo okwandisa ugesi sezitokisi, kuyashesha ukukhula kwabo kanye kwamangqamuzana, isisindo somzimba kanye ukusheshisa izinqubo umzimba. Omunye abameleli leli qembu izidakamizwa "Riboxinum".

izici kwemithi zomuthi

Ukulungiselela "Riboxinum" limelela umkhiqizo Anabolic okwelapha, umphumela eyinhloko okuyinto iqondiswa ukwandisa izicubu ukumelana nezimo hypoxia. Njengoba eyandulela ka triphosphate adenosine, "Riboxinum" abathintekayo ezinqutsheni cleavage glucose ngaphakathi kwengqamuzana futhi, ngenxa yalokho, ukwakheka triphosphate adenosine, okuyinto enkulu iseli amandla substrate. Ngenxa yalokhu umphumela "Riboxinum" uzabalaza umphumela anti-hypoxic ngokuya kwehle okuqukethwe ATP.

Steroid umphumela "riboksin" owabonakaliswa anda umzimba izinqubo ezihilela pyruvic acid futhi kusebenze xanthine dehydrogenase. Ngenxa miphumela "Riboksin" unethonya elihle inkambo imiphumela umzimba ngaphakathi kwamaseli womuntu, ukuthuthukisa amandla abo asinikeza operation evamile.

Lapho wadalula myocardium "Riboxinum" lithuthukise myocardiocytes, waba nomthelela ekwandeni okwengeziwe okuphelele ukuphumula yabo (okwandisa phosphorylation i izibopho actin-myosin) futhi oyenza izinqubo okuzivuselela e myocardium.

Ngokuya izinqubo pharmacokinetic "Riboksin" fed ngokuphelele phakathi kwegazi kakade mafutha anciphisa isikhala esingaphakathi yokusetshenziswa pheshana emathunjini. Ukuze imizila parenteral yokuphathwa (i.v.) "Riboxinum" ngokwanele ngokushesha ukusatshalaliswa izicubu ukudlula izigaba okwalandela kumaseli umzimba kwesibindi, lapho eqhekeza egcwele. Excretion of metabolites unmetabolized kanye nama-molecule izidakamizwa kwenzeka ogxile emchamweni, futhi ingxenye encane lisuselwa indle kanye Bile.

izinkomba

Izidakamizwa "Riboksin" wabonisa ekwelapheni isifo senhliziyo, kuhlanganise nalezo ekwelapheni post-infarction uthi. Umuthi inomphumela omuhle zokwelapha ekwelapheni uthi isigqi kanye conduction thuthuva, ukweqisa izidakamizwa unamasu inhliziyo glycosides, ekwelapheni ukukhubazeka morphological imisipha yenhliziyo, okubangela zangokwasemuva zezinhlelo anda umthwalo ngokomzimba, noma ngemuva zezifo ezithathelwanayo namakhambi ukuvuvukala.

"Riboxinum" kuboniswe yokwelapha izifo kohlelo hepatobiliary, nokuvimbela izifo kohlelo igazi ekulungiseleleni ebulilini ionizing emisebeni. Ngo umkhuba amehlo, ukusetshenziswa "riboksin" kunilungele ngesikhathi evulekile-engela glaucoma.

"Riboksin": yokusetshenziswa, analogs

Lapho usebenzisa i-sefomu tablet ye umuthi ukuba banamathele lezi zincomo. Kubantu abadala, umthamo wansuku zonke zomuthi zingaba phakathi 0.6 kuya 2.4 amagremu. Ngokuvamile, umthamo is kushintshwe ngamunye, kanye umthamo wansuku zonke sehlukaniswe ngemithamo eziningana usuku lonke. Khomba ifomu tablet kufanele kube umthamo ubuncane, futhi kuphela uma umthamo ubuncane ngokuvamile ikubekezelele nesineke, ngemva kwezinsuku ezingu-2-3 ekutheni kube nokubuyisana. Isikhathi yokwelapha kufanele kube kusuka 1 kuya 3 izinyanga.

Ngo ekuphathweni parenteral, isixazululo 2% "Riboxinum" buhlanjululwe 250 ml we nosawoti sodium chloride noma glucose. I ukumnika Kwenziwa kancane ngesilinganiso esingamaphesenti 40-60 amathonsi ngomzuzu.

analogs engeziwe nge Isikali efanayo kufanele kuqashelwe, "Inosine" futhi "Ribozin", okuzoxoxwa ngezansi.

Izimo izidakamizwa

Izimo ukunikeza ukuzwela eyengeziwe eyodwa noma ngaphezulu yezingxenye izidakamizwa, sifo kanye namazinga angcono uric acid-plasma yegazi. Ngokucophelela okukhulu kufanele libekwe "Riboksin" futhi Analogue "riboksin" "Inosine" iziguli ezine ukwehluleka kwezinso umsebenzi excretory.

side effects

Ngokuvamile, izidakamizwa babekezelelwa kahle. Phakathi kwalabo abaye bakubona ukuzwela kwabaningi izidakamizwa kungabonakala nasemkhakheni kusukela isikhumba yokungezwani komzimba. On the ingxenye esimiso senhliziyo nemithambo yegazi kungadala palpitations, kukhuphuke blood pressure, ubuthakathaka.

Esimweni lapho isiguli ethola 'Riboksin "kuphawula okungenhla side effects, kumele uxhumane nodokotela wakho futhi uyeke ukuthatha izidakamizwa.

imiyalelo Special ukuthola

Njengoba "Riboxinum" futhi metabolites zalo excreted ngokuyinhloko izinso, ke asifanele ukusetshenziswa kwezidakamizwa ebukhoneni ukwehluleka kwezinso. Ukusetshenziswa kwalesi izidakamizwa kungavunyelwa kuphela esimweni lapho izinzuzo kulindeleke zomuthi okukhulu naphezu kwengozi engase ivele yokusetshenziswa kwawo. Hambisana imithetho efanayo ukuqokwa izidakamizwa kwabesifazane abakhulelwe kanye lactating.

Nakubukwa umtselela "riboksin" ezingeni uric acid -plasma yegazi ngesikhathi yokwelapha Kunconywa ukuqapha yayo njalo ukuze uvimbele okuvela hyperuricemia.

Ubuthi futhi izidakamizwa ukweqisa izidakamizwa

Uma ekutholeni ebulilini nomuthi wayebaphathele izinyathelo jikelele okuhloswe ngazo ukunciphisa izidakamizwa ngokufaka ekusakazeni igazi. Endabeni ka izimpawu ubuthi - yokwelapha lingaze. Lapho komzimba, ukwelapha ebulala kuyaphumelela.

"Riboksin": nozakwabo

Kuze kube manje, emakethe ezithaka imithi akekho noyedwa Analogue "riboksin" mode Anabolic yesenzo. Kulokhu, kukhona kokubili analogs equkethe nezinye isithako esebenzayo, kanye omqondofana ephelele izidakamizwa, babe ukubunjwa yabo efana isithako esebenzayo.

"Inosine" ingase ifane ngalokho ekushoyo kanye analog ngokugcwele "Riboxinum" kwezokuphatha esicutshini. Enkabeni yalo, umuthi engathatha okuphelele "riboksin" nazo zonke izinkomba zayo kanye contraindications. Enye elifanayo kubhekwe izidakamizwa - "Ribonozin". Lokhu ukulungiselela iqukethe isithako esebenzayo, umuthi ezifanayo "Riboksin" ukubunjwa yayo. Analogue izingane isiraphu - umuthi ngokuthi "Mildronat". Ubuye ikhono ukunikeza amandla homeostasis cishe yonke kumaseli emzimbeni.

Uma sicabangela iqembu izidakamizwa ezingekho steroidal Anabolic, singakwazi ukuhlukanisa analogs ezinjalo "Riboxinum" amaphilisi "Methyluracil" kanye potassium orotate. Le mishanguzo, nakuba zingezikaJehova amaqembu ehlukene kwemithi, Nokho, bayakwazi nethonya umphumela Anabolic. Ngokuvamile, lo mphumela kungenxa ukukhuthazwa izinqubo umzimba wonke kwamangqamuzana nezicubu zomzimba.

Ukuqhathanisa ne izidakamizwa "Riboksin" nozakwabo isizukulwane esisha, siphawula ukuthi abe nekghono ephakeme nemiphumela zokwelapha. Ummeleli uyakufanelekela leli qembu "Citoflavin". Lokhu Analogue "riboksin" Ngaphezu yemiphumela cytoprotective kanye antioxidant futhi emnandi umphumela elinamandla izinzwa ingqondo.

isiphetho

izidakamizwa steroid - izidakamizwa iqembu ezibanzi ezahlukene isakhiwo sazo sekhemikhali. Kuye inhloso ohlela ukuzisebenzisa, ungakhetha "Riboksin" izidakamizwa analogue, noma ngonanzelelo iqembu steroid. Qaphela ukuthi it is hhayi Kunconywa isicelo ezimele le mithi. Kuphela onguchwepheshe oqeqeshiwe kungasiza Ukukhetha izidakamizwa.

Similar articles

 

 

 

 

Trending Now

 

 

 

 

Newest

Copyright © 2018 zu.unansea.com. Theme powered by WordPress.