ImpiloAmalungiselelo

Eye lehla "Lyuksfen": yokusetshenziswa, analogs kanye nokubuyekeza

Indlela okufanele ngiyisebenzise ngeso lehla "Lyuksfen"? Imiyalelo yalesi izidakamizwa uzobe zichazwe ngokuningiliziwe ngezansi. Futhi kule materials sihloko sinikeza ulwazi ngalokho kuyadingeka, wathi izindlela, kuze kufike kuyaphumelela ukuthi unakho nozakwabo.

Ukuma kanye nokwakheka

Equkethe izidakamizwa ngokuthi "Lyuksfen" (iso amaconsi)? Umhlahlandlela ugomela ngokuthi ukwakheka kwe-nomuthi kuhlanganisa brimonidine tartrate (isithako esebenzayo), kanye izakhi ukwesekwa ngesimo benzalkonium chloride, i utshwala we chloride polyvinyl, sodium citrate dihydrate, citric acid monohydrate, hydrochloric acid, amanzi kanye sodium hydroxide.

Kulaba izimali itholakale ukudayiselwa ngesimo esobala ngeso lehla umbala ogqamile ephuzi. Isixazululo yafakwa amabhodlela weThrojani eyenziwe polyethylene, amakhadibhodi iphakethe, ngokulandelana.

Yezemithi kwezidakamizwa wendawo

Indlela yokufaka isicelo ngeso lehla "Lyuksfen"? Umhlahlandlela ibika ukuthi ukuphumelela izidakamizwa ngokuphelele ngenxa isithako yayo asebenzayo. Brimonidine kuyinto agonist ukukhetha alpha-2-adrenoceptors.

Ngemva kokufaka 0.2% isixazululo Pressure ukunciphisa (intraocular) cishe 10-11 mm HG. Art. Umthelela esiphezulu zomuthi kokubuyekezwa amanothi ngemuva kwamahora amabili. Kulokhu, kusebenta oqabulayo imithi nezokusigcoba siyenzeka amahora 12.

Ngokusho ochwepheshe, brimonidine has a indlela ombaxambili senzo. Ngeke nje kuphela ukwehlisa ingcindezi (intraocular) ngokunciphisa inani synthesis uketshezi intraocular, kodwa futhi ukuthuthukisa outflow uveoscleral.

isixazululo kinetics ngeso

Iziphi izici kinetic babe ngeso lehla "Lyuksfen"? Umhlahlandlela ithi ngemva instillation of 0.2% isixazululo izidakamizwa kabili ngosuku izinsuku ezingu-10, emakamu yayo egazini liphansi kakhulu (mayelana 0,06 ng / ml).

Uma ufaka nomuthi kubhekwe lokuhlushwa yayo eliphakeme esegazini kufinyelelwa ngemizuzu engaba ngu-30-95. Brimonidine isigamu zokuphila kwabantu ezivela enkulu yomzimba womuntu yakhiwa cishe amahora amabili.

ukumuncwa lefundo isithako esebenzayo kuyinto amathonsi kancane. Wendawo isicelo uxhumano amaprotheni igazi imayelana 29%.

Umzimba izidakamizwa wenziwa ngokuyinhloko isibindi.

Isici esebenzayo yalesi izidakamizwa futhi metabolites zalo excreted ngokusebenzisa nezinso.

Izinkomba ukusetshenziswa amathonsi

Ingabe uyazi ukuthi kuzinjongo iziguli kuyabekwa ngeso lehla "Lyuksfen", analogue zazo kukhonjisiwe ngezansi? Ngokusho imiyalelo, le nomuthi kuboniswa for ekwelapheni izifo ezifana:

  • ocular (ukusetshenziswa njengoba monotherapy futhi lihambisana namanye amanxusa ukuthi kuncishiswe ingcindezi intraocular);
  • evulekile-engela glaucoma.

Uvala ukusetshenziswa imithi nezokusigcoba

Ngaphansi akukho Izimo Awukwazi ukusebenzisa iso lehla "Lyuksfen"? Ukufundiswa uthi izidakamizwa okukhulunywa kungavunyelwe yokunika kulezi zimo ezilandelayo:

  • ngenkathi ibele ingane;
  • ukwelashwa ngesikhathi esifanayo ne-tricyclic antidepressant futhi mao inhibitor;
  • ngaphansi kweminyaka eyi-2;
  • hypersensitivity kuya izidakamizwa izidakamizwa.

isabelo ngokucophelela

Drops "Lyuksfen", okuyinto Izibuyekezo zingaphezu omuhle, ebekiwe ngokuqapha ukuze abantu thromboangiitis obliterans, ifomu engazinzile, ezinzima noma engalawuliwe yokuthola izifo eziphathelene nenhliziyo, esingamahlalakhona senhliziyo noma i-cerebral, hypotension orthostatic, isifo Raynaud kanye nokucindezeleka. Futhi ebekiwe ngokuqapha kwabancane kanye ukungasebenzi kwesibindi noma izinso.

Eye lehla "Lyuksfen": yokusetshenziswa

Lo mkhiqizo senzelwe ukusetshenziswa ngezihloko ezihlukene kuphela. Ukuze ekwelapheni izifo amehlo ezifana nomfutho wegazi ophezulu ocular futhi evulekile-engela ukufiphala le nomuthi lwagxiliswa izitho ezibukwayo 1 iconsi kabili ngosuku. Isikhathi ukwelashwa nge leli thuluzi kuchazwa kuphela nguchwepheshe, okungukuthi, kudokotela wezifo zamehlo.

Izenzo-uhlamvu

Kungabangela abantu basabele ngendlela embi ngeso lehla "Lyuksfen"? Nobufakazi bathi ngokumelene isizinda izidakamizwa ngokuvamile sibhekana nemiphumela elandelayo enqabayo:

  • hyperemia conjunctival, conjunctivitis nomzimba, amehlo silume ulwelwesi lwamafinyila kanye isikhumba amajwabu amehlo;
  • folliculosis conjunctiva samehlo, ukuncinza, conjunctivitis follicular, blepharitis, ukusabela wendawo iguliswa we ulwelwesi lwamafinyila kwezitho ezibukwayo, kuhlanganise keratoconjunctivitis;
  • osenyameni lwamafinyila emehlweni, blepharoconjunctivitis, ukopha conjunctival, ukuzwakala kahle ngombono, ubuhlungu nokuvuvukala amajwabu amehlo, ale nkinga, keratitis, edema conjunctival, umonakalo ubudala, conjunctivitis, amehlo zamanzi, epiphora, keratopathy zinamabala, ukucasuka bese we iso;
  • photosensitivity, ububomvu amajwabu amehlo, ukulahlekelwa obusebenzayo yomzimba Vitreous, nomzimba angaphandle ukuzwa kwezitho ezibukwayo, ukulahlekelwa emkhakheni umbono, angaboni kahle, ukopha emzimbeni Vitreous, opacities elintantayo emzimbeni Vitreous;
  • anda blood pressure, ukuguguleka corneal, ikhanda, ibhali, ukuqwasha, kunciphisa umfutho wegazi, ukozela, ukucinana kwemigudu yokuphefumula, isiyezi;
  • ukukhwehlela, dyspepsia, ezomile nolwelwesi lwamafinyila ikhala, ukuqubuka, ukuphelelwa umoya lapho belele, iphika;
  • kome umlomo, umkhuhlane syndrome, rhinitis, nezifo ezithelelwanayo angase azithole (izinkinga zokuphefumula futhi Ukugodola), sinusitis;
  • hypercholesterolemia, asthenia, ukusabela jikelele umzimba uxabane nawo, ukukhathala, bradycardia, izinguquko ukunambitheka emizweni, hypotonia kwemisipha, hypothermia;
  • iritis, ukucindezeleka keratoconjunctivitis, tachycardia, amajaqamba, isicanucanu, ukusabela isikhumba bendawo, kuhlanganise zokuzikhukhumeza ebusweni, erythema, amawala, ukulunywa futhi isikhumba vasodilation semithambo ubudala.

Ukweqisa izidakamizwa imithi ukuze iso

Kwenzekani uma uthatha ku ngeso lehla "Lyuksfen"? ochwepheshe lezivakashi bathi uma kokungenisa ngephutha yesixazululo, izimpawu ezilandelayo ukweqisa izidakamizwa ahlanganisa ukozela, CNS ukudangala, ukungakuthandi nokucindezeleka ukwazi, bradycardia, kunciphisa umfutho wegazi, cyanosis kwesikhumba, ukwehla kwezinga lokushisa komzimba, futhi elele singathatha.

Lapho izimpawu esinjalo isiguli sidinga bangisekela yokwelapha lingaze, kanye nokuqapha zokuphefumula ipheshana isimiso.

Ukuxhumana nezinye izidakamizwa

Kungenzeka yini ukuba sihlanganise namanye amaconsi "Lyuksfen" izindlela? Yokusetshenziswa lithi brimonidine at lokuhlushwa 2 mg / ml ithuthukisa kalula isenzo izidakamizwa ezithinta isimiso sezinzwa esiyinhloko (lapha zihlanganisa utshwala, opioids, barbiturates, imithi ebulala izinzwa, futhi sedatives).

Kuyadingeka ukuba unakekele ekhethekile ngenkathi izidakamizwa kungathinta ukumuncwa futhi metabolization adrenaline futhi noradrenaline nezinye ama biogenic (isib methylphenidate, chlorpromazine, reserpine).

Kwezinye izimo, ngemva isicelo sale nekhambi lokuhlushwa 2 mg / ml iziguli zehle ngo okuncane wegazi. Kule ndaba kufanele uqaphele ikakhulukazi ngokusebezisa parallel imithi antihypertensive noma izidakamizwa okuqondene iqembu glycosides inhliziyo.

Ibele nokukhulelwa

Kungenzeka yini ukuba ngabele imithi abakhulelwe kanye lactating abesifazane "Lyuksfen" (ngeso amaconsi)? Ukufundiswa uthi ucwaningo ukuphumelela nokuphepha yokusebenzisa lolu imithi ezingazange iqhutshwe leli qembu labantu. Kufanele kuqashelwe ukuthi ngokuhamba ukulinga izilwane ukusetshenziswa endawo brimonidine ayimlethelanga yikuphi ukuphulwa wokukhula kwengane esiswini. Futhi akukho ulwazi ngqo mayelana Ukungena izidakamizwa ubisi lwebele uma isicelo ihlelwe ngokulandelana kwezihloko. Kulokhu, ingozi is hhayi iqedwe ngokuphelele.

ulwazi oluthile

contact lens kumelwe kususwe ngaphambi kokusebenzisa eyedrops. Isikhawu esiphakathi isicelo zomuthi futhi ufaka lens kumele okungenani ibe ¼ ihora.

Kusukela nomuthi kubhekwe kungabangela ukozela noma ukukhathala, futhi yehlise acuity ezibukwayo, ngesikhathi yokwelapha izidakamizwa kufanele uyeke ukushayela izimoto kanye nokugcinwa ezihambayo eziyingozi izingxenye.

Imigomo nemibandela isitoreji, leli holidi izidakamizwa

Eye lehla "Lyuksfen" akhishwa Pharmacy ngaphandle udokotela. Iqukethe isidakamizwa enjalo kufanele ibe lokushisa akukho ephakeme kuka-degree 25, esikhundleni kude nezingane.

Impilo yesixazululo uneminyaka engu 2 kusukela usuku ukwakhiwa. Ngemva kokuvula isitsha, le nkathi kuyehla kube amasonto 4.

amalungiselelo Okufanayo futhi omqondofana

Manje uyazi ukuthi lokhu yisisombululo bendawo ukuba iso, njengoba "Lyuksfen". Imiyalelo analogs ka kulo muthi okuxoxwe ngazo kulesi sihloko.

Uma izidakamizwa wathi kuhlulekile ukuthenga, kungashiwo indawo ngezindlela ezifanayo njenge "Clonidine" (iso amaconsi). Ngokusho indlela yayo yesenzo yalesi izidakamizwa liseduze kakhulu ngale ndaba. Ngaphezu kwalokho, kungokwalabo iqeqebana efanayo kwemithi.

Ngokuphathelene omqondofana ukuthi uyifunda izindlela ezifana "Alfagan P" futhi "Alfabrim" (izixazululo amehlo). Le mithi kufanele isithako efanayo esebenzayo.

umthengi Izibuyekezo

Ngaphambi kokuthenga la noma ezinye izidakamizwa, abantu abaningi ufunde mayelana imibono yabo abathengi. Kufanele kuqashelwe ukuthi ukubuyekezwa ngeso lehla "Lyuksfen" kukhona abaningi kangaka. Iningi lawo abantu okuhle. Labo iziguli "Lyuksfen" waqokwa ophthalmologist, bame kwelokuthi lokhu kuyinto esebenza kahle kakhulu futhi ngempumelelo izidakamizwa. isicelo sayo efanele futhi ifike ngesikhathi ikhuthaza ekwelapheni izifo ezifana nomfutho wegazi ophezulu ocular futhi evulekile-engela glaucoma. Kumele ngokushesha zaphawula ukuthi le nomuthi singasetshenziswa hhayi nje njengomuntu monotherapy kodwa futhi lihambisana namanye izidakamizwa ukuze iso.

Ngeshwa, kuzo zonke izibuyekezo kule nomuthi zingatholakala nemibi okuthunyelwe. Iningi lazo zixhumene ukuthuthukiswa amathuba okuba nemiphumela engemihle. I ngokuvamile kubonakala khona ukusabela ezingezinhle yilezi: ukuqubuka ku Isivalo, ububomvu samehlo, ukukhathala, komzimba, kanye nezinye zendawo. Ngaphansi kokuqondisa ezifana side effects, ochwepheshe batusa ukuba enqabe ukwelashwa ngendlela eyengeziwe. Kulokhu, isiguli kungcono yokunika ehlukile, imithi ephephile.

Njengoba for izindleko iso amaconsi, e ezahlukene ekhemisi ngamaketanga kwehlukile. Nokho, isilinganiso senani umuthi ruble 350-370. Ezinye iziguli zithi droplet okukhulunywa izindleko ezeqile, kodwa abanye kwamukeleka ngempela.

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