ImpiloAmalungiselelo

"Flutamide": yokusetshenziswa, incazelo izidakamizwa, analogue nama-side effects

"Flutamide" ingenye elwa ne-androgen futhi esetshenziselwa izimpawu ukuqedwa androgenization. It has ikhono kukhawulwe umzimba hormone androgenic luqhubeke ngempumelelo umphumela wawo izitho abadinga ukwelashwa. Injongo eyinhloko izidakamizwa - nokucindezela hormone wesilisa, ngempumuzo izifo zibangelwa ngokweqile ke.

izakhiwo kwemithi

Umuthi 'flutamide-250 "okungukuthi ezisetshenziswa ekwelapheni abesifazane nabantu izimpawu okhushuliwe testosterone ukukhiqizwa ethintekile esibi imiphumela kuwukubonakaliswa le hormone. izidakamizwa Non-steroidal zivimbela biosynthesis ka androgens kanye uketshezi of nezindlala kuyehla ukukhiqizwa gonadotropin nokwehlisa lokuhlushwa androgens molecule asebenzayo. Umuthi oyenza izinqubo umzimba, kuthuthukisa umzimba umsebenzi ekususweni hormone ngokweqile excreted.

Libhekisela eqenjini non-steroidal izidakamizwa antagonizes 5-a-reductase. Ukwamukelwa "flutamide" Akunamthelela lapho kuvezwa gonadotropin ku pituitary indlala futhi kunciphisa gonadotrophic umsebenzi.

Izinkomba for Ukwamukelwa

Ukuphumelela ukuphathwa kuletha umphumela eziyinkimbinkimbi ku inqubo ekunciphiseni izinga hormone asebenzayo. Lokhu kwakwenziwa ngayiphi injongo wasebenzisa "flutamide"? Yokusetshenziswa imibukiso nokwehla, futhi kamuva androgenization unyathela amabhuleki inqubo.

Ngenxa ukwandisa umkhiqizo androgen luphakanyiswa umsebenzi enzyme 5-α-, ehilelekile kabusha isikhumba kanye yokwamukela yayo ikhuthaza luvelo la ma-hormone. uyiqala kanjalo nokuthuthukiswa hirsutism idiopathic abadinga ukwelashwa.

Kuze kube muva nje uye wamiswa ekwelapheni Hyperplasia Prostatic ezingabantu, kodwa hhayi kangako kudala Kwakubonakalisiwe nomphumela walo omuhle ngoba impatho ngempumelelo ezinye izifo ezihlasela abesifazane. Hirsutism, Alopecia "flutamide" kwabesifazane ngesikhathi kwansuku reception izinyanga ezintathu kwanele ukunciphisa ngempumelelo igazi amazinga anda hormone wesilisa, futhi lezi zifo iphelelwa ngobubi bawo.

Izifo lapho kuboniswa ngokuthatha izidakamizwa

  • umdlavuza wendlala yabesilisa ukusabalala metastases ezingabantu.
  • Hirsutism futhi Alopecia kwabesifazane.
  • Lapho kuhlinzwa castration babantu.
  • Lapho iziyaluyalu hormone nge izimpawu induna.
  • Ngo kwesisu noma ukungakwazi nje ebamba isisu.

The main izinkomba nezimpawu ezisikisela i overabundance kwe-testosterone emzimbeni. Ngo abesifazane, okweqile izinwele umzimba wesilisa pattern impandla, iziyaluyalu kokuya esikhathini nokunye. D. Kukhona futhi hormone umzimba nge izimpawu esicashile ezifana anovulation, hypoplasia kwesibeletho kanye nezindlala mammary.

Ukuze udokotela uphethwe i olunembile uqoka kokuxilongwa ezengeziwe, okusho uthole ukucwaningwa okuningiliziwe kokulandisa ukuhlolwa igazi isimo izinga lama-hormone ezihlukahlukene emzimbeni.

ukusetshenziswa Independent zomuthi, ngaphandle ngokulandela isincomo udokotela ukuba khona, kungabangela umonakalo ongalungiseki impilo. Linqume ukwelashwa kufanele kube ngokuqinile udokotela!

reception Izici

Ukuze ukulungiselela "flutamide" imfundo manual kubonisa ekuzuzweni kwemiPhumela esiphezulu lokuhlushwa igazi 2-3 amahora emva yokwemukelwa, lubonise okusheshayo absorbability izidakamizwa emathunjini. Ingxenye-ukuphila cishe 5-6 amahora emchamweni, futhi kamuva, ngemva kwamahora angu-8-9, amasalela kuyinto okukhiphayo. zizalela Quality incike yobudala lesiguli kanye kwezempilo jikelele.

Izifo nge nezimpawu androgenization abesifazane zidinga abathile ukwelashwa. Icacisa ngokwezinga, kanzima indawo izindawo inkinga nezinye izinto ukuthonya enquma izidakamizwa, ngokuvamile "flutamide" inikezwa complex reception. Yokusetshenziswa libonisa reception triply emini omunye capsule, ukugcina ngezikhathi ezithile. I nsuku zonke umthamo 750 mg, ubuncane isikhathi sokwelashwa okungukuthi kwamasonto ayisithupha.

izimpawu yokwelapha ngenxa yokuqukethwe okwandisiwe androgens kufanele kuhlanganiswe neminye imithi ethile izakhiwo anti-androgenic. Ngokuvamile ekuhlanganisweni esimisiwe 'Dexamethasone "," Prednisolone "nezinye izinto ezithwala ngama-corticosteroid. Sebenzisa futhi esithobayo ukwelashwa ukusekela nezindaba zempilo yengqondo kweziguli simtomov nezisobala kubangelwa isiphithiphithi hormone.

Ngisho nalapho engekho izimpawu ngaphambili ukhathazeke ukukhansela izidakamizwa wedwa akunconyelwe lokhu kufanele ubuze endocrinology, ethungatha ukuthuthukiswa lesi sifo. Kumele esiqinile nokulandela yonke imithetho ephathelene kadokotela. Uma nganoma isiphi isizathu ukuqokwa ukuthi uphuthelwe amaphilisi, akufanele uthathe elandelayo ezimbili, futhi nje ugcine reception evamile. Yeqa izidakamizwa akuyona kulimaza njengokungenisa olulodwa ethola umthamo double.

ukukhululwa Ifomu

Ikhishwa ngesimo amaphilisi noma amaphilisi ifilimu-camera. Ifanele reception ngomlomo. Ngempumelelo izidakamizwa esebenzayo - flutamide 250 mg.

Amakhemini "flutamide" UYADAYISWA kuphela kadokotela.

Gcina endaweni epholile, endaweni eyomile aphume kude nezingane.

Ukukhiqiza - Orion Corporation, inkampani eyenza imithi (Finland).

On the "flutamide" Intengo kusuka 1798 kuya ruble 1968 iphakethe ngasinye (amaphilisi 84).

Izimo

Njengoba kuboniswe, isipiliyoni ekwelapheni abesifazane eside ngokwanele, ngokuyisisekelo kumayelana ukungaqiniseki nolwazi side effects kanye nemiphumela emibi isibindi. Ngakho-ke, naphezu okusezingeni eliphezulu lempumelelo izidakamizwa kumele kusetshenziswe ngokuqapha, okulandelayo iseluleko odokotela.

  • Okunqatshelwe reception "flutamide" iziguli ezine yezifo yegilo indlala, isibindi noma izinso.
  • Hypersensitivity emuthini "Flutamide."
  • Izimo e iziyaluyalu izinso, pancreas.
  • Okumele kuqashelwe ukuthatha e propensity ukwakha amahlule iziyaluyalu yisimiso senhliziyo nemithambo yegazi.

Ukuxhumana nezinye izidakamizwa

Ngaphambi kokusebenzisa umkhiqizo letiphakanyisiwe ukwazisa udokotela okuyinto nemithi zithathwa njalo. Udokotela kumele ibhekelele izinto eziphathelene amavithamini isikhalazo, Izithako zokudla, kuze reception carbon isebenze.

  • "Flutamide" ngenkathi ke ukusetshenziswa neminye imithi ikwazi potentiate antiogulyantov kudinga efanele Isikali ukubala, ikhumbula nokuxhumana.
  • Ukubhema kanye notshwala ingase futhi guqula isenzo izidakamizwa emzimbeni. Ngesikhathi reception kuyoba okunengqondo Sinike kuze ezimbi imikhuba.
  • Mayelana ezikhona igazi izifo udokotela futhi kufanele unolwazi.
  • Uma uhlela ukukhulelwa, qiniseka ukuthi ubona udokotela ngoba reception olwengeziwe.
  • Umbiko ka-iguliswa ukusabela emithini, uma zikhona, futhi lokhu okungukuthi kahle aziwayo.

ukweqisa izidakamizwa

Uma ngephutha wathatha umthamo enkulu amaphilisi "flutamide," kubalulekile lavage esiswini kanye ukwelashwa esibhedlela noma "ambulensi". Imiphumela ukweqisa izidakamizwa kungabangela unomphela ngokweqile isithuthukisi abacindezela i-hormone noma gonadotrophin ngokuphelele nse ukukhiqizwa, ehamba phambili kwesinye isifo. Ngakho-ke akuyona ukuhambisana kudingekile nemithetho, ukuthatha "flutamide" yokusetshenziswa libhekisela ekuhambisaneni umthamo kanye nodokotela.

isicinganani

Ngemva kwesikhathi eside ukusetshenziswa indoda kungathola izimpawu of gynecomastia, ubuhlungu webele, nokugcinwa uketshezi.

Uma asho into elandelayo, okungaba izimo ezilula bokuphila, umuthi kufanele kuxoxwe nodokotela wakho, ikakhulukazi uma ngaphambi lena kwakungeyona.

Izimpawu amathuba okuba nemiphumela engemihle

  • Ukuqunjelwa.
  • Ukwephula iphango.
  • Ukwehla libido.
  • Wamabele ukukhulisa ezingabantu.
  • uthi futhi bacindezeleke.
  • Ukwephula ubuthongo futhi sihlale siphapheme.
  • Ukuvuvukala.
  • Izinguquko ngombala umchamo.
  • Ukukhathala.

Ukusabela Esibi - ukungasebenzisi, kodwa lezi zimpawu ukwazisa kangcono udokotela kungase kudingeke ushintshe okuthile indlela athole impatho noma uyeke ukuthatha imithi.

analogs

Antiandrogens - iqembu izidakamizwa kokuba impahla abacindezela isizukulwane ngokweqile progesterone okubangela thuthuva lizwakale abanempilo lesiguli. By "flutamide" esifanayo imithi ezilandelayo ze-non-steroidal akunakubangelwa phezu izakhiwo kanye nokusungulwa:

  • "Cyproterone" - ukulungiswa obujwayelekile iqembu progestogens nge antigonadotropnym umsebenzi.
  • "Spironolactone" ( "Veroshpiron"). Eyesibili izidakamizwa ethandwa kakhulu, "flutamide" izimiso replaceable ithonya iyafana, mhlawumbe ngisho izakhamuzi zaseBosnia zifana.

Ngaphambi kokuqala yokwamukela noma yimuphi iqembu unikezwa zomuthi ukuqinisekisa ukuthi umthombo isifo singakabi ahlobene ekukhulelweni lwesimila. Kuthatha ukulungiselelwa ngokucophelela ukuze indlela ekwelapheni hyperandrogenism, ukwemukele Izimo akhawunti kanye izici ngazinye esigulini ngasinye. Kubalulekile edilini ngesikhathi udokotela ukuchaza ngokuningiliziwe izimpawu zokubonisa sifo, okuthiwa izifo ezikhona, ikakhulukazi uma zihlotshaniswa kokusebenza kwesibindi, indlela kuphela udokotela Ungakhetha ukwelashwa ngoludala ngokuhlanganyela "flutamide."

Izibuyekezo

Kafushane ukhulume izimpendulo mayelana ukuphumelela izidakamizwa "Flutamide." Izibuyekezo zibe khona kungaxoxwa ngazo abantu abaye baphathwa. Ngo abesifazane abaphethwe izimpawu of hirsutism, lo ukuzinza izinwele zikhula zibheke ngakhona. I nezindlala sebaceous esikhumbeni, okubangela induna, futhi waphinde waba nemisebenzi yayo evamile.

Kuye kwaba nezenzakalo ukuthi akuzona kakhulu eziwusizo "flutamide" Izibuyekezo akazange qinisekisa elikhethekile inzuzo ngokuthola eyamukelayo, maningi amathuba okuthi ngenxa elingalungile ukuxilongwa noma amaphutha isicelo. Ezinye iziguli Ungasingenisi inkambo eside ukwelashwa kuze kube sekupheleni intengo izidakamizwa, kulesi simo, ungakwazi bonana nodokotela wakho kuqala resort kunemifuziselo eshibhile, ukuze singathwesi phela yokwelapha. On the "flutamide" intengo okungukuthi ngempela high futhi udinga ukuthatha lokhu ku-akhawunti, ukuphathwa okungukuthi ngempela ezinde kuzodinga zezimali ngokukhwabanisa.

Izixwayiso

Lapho eziyinkimbinkimbi ukuphathwa izinsuku ezintathu ngaphambi isicelo GnRH agonist kufanele kuthathwe "flutamide" ukuze unciphise amathuba okuba nemiphumela engemihle. Lapho isibindi ukwehluleka ukwelashwa kuboniswa kuphela uma okungukuthi kuphela indlela uzimise- le nkinga. Kumele kwenziwe laboratory Ukutadisha umsebenzi kwesibindi. Kube nokwenyuka abanye e isibindi lapho ithola "flutamide," kodwa ngemuva kokuhoxiswa iba isinqumo evamile. Lapho izimpawu okungafunwa Kunconywa ekususweni izidakamizwa.

ukuhlolwa Ifanele laboratory ukuhlola umsebenzi ukuhlolwa isibindi kufanele kwenziwe esigulini ngasinye kanye ngenyanga phakathi nezinsuku zokuqala izinyanga 4, bese ngezikhathi ezithile noma ngesikhathi ukuthuthukiswa izimpawu zokuqala ngalesi sifo umsebenzi hepatic (ukulunywa, umchamo onombala, ukulahlekelwa okusimeme esesuthi, jaundice, amaphaphu ilungelo quadrant engenhla). Ukuze uthole eside isikhathi Ukwelapha amadoda e ukungabikho amakhemikhali noma kuhlinzwa castration kufanele njalo kuhlolelwe isidoda ukulondolozwa wenzalo.

On the subject of ukushayela imoto futhi izindlela zokuphatha izifundo sezenziwe. Kodwa uma unanoma iluphi uhlobo izimpawu njengokuba nesiyezi noma ikhanda, kungcono ukuthatha izingozi futhi hhayi ukuhlala beshayela.

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