ImpiloAmalungiselelo

"Proflosin": yokusetshenziswa, ngempela

Kungani akunikeze imithi "Proflosin"? Yokusetshenziswa zomuthi, imiphumela engemihle, contra-izinkomba, futhi uzobe wachaza ngokuningiliziwe kulesi sihloko. Ngaphezu kwalokho, sizokutshela ukuthi uma unayo le imithi analogs, ukuthi kubiza malini futhi abakushoyo ngaye iziguli.

Khipha ifomu kanye nokwakheka

kusho "Proflosin" ithengiswe kunoma yiluphi uhlobo? Yokusetshenziswa yazisa ukuthi lokhu izidakamizwa itholakala ifomu capsule ekukhishweni ukushintshwa. nomuthi Okubukwe iqukethe element asebenzayo ezifana tamsulosin hydrochloride. It Ubuye adjuvants njengoba triethyl citrate, microcrystalline cellulose, talc, kanye copolymer ka ETHYL acrylate futhi methacrylic acid.

izici kwemithi

izidakamizwa "Proflosin" Isebenza kanjani? Imiyalelo isicelo uthi ketshezi asebenzayo kubhekwa indlela uyakwazi ngokuncintisana futhi ngokukhetha ukuvimba ama-receptor α1A-adrenergic (postsynaptic) ezisesandleni imisipha abushelelezi esinyeni entanyeni, wendlala indlala futhi urethra Prostatic. ukuchayeka okunjalo kuholela ekuphikeni nokuncipha bushelelezi imisipha ithoni, esiza ukuthuthukisa umchamo ukugeleza.

Asinakusho ukuthi α-adrenoceptor blocker ukunciphisa umfutho wegazi ngenxa ukwehla ukumelana semithambo (neuropathy).

izakhiwo pharmacokinetic

izidakamizwa "Proflosin" Long noma ugxile? Iziyalezo yokusetshenziswa uthi ngemuva kokuthola amaphilisi tamsulosin ngaphakathi kahle ngokushesha ugxile kusukela pheshana emathunjini. Nokho, ukumuncwa yayo siyehla kancane emva kokudla. Ngo umthamo owodwa we-nomuthi ngezilinganiso ka 0.4 mg emakamu eliphezulu kakhulu izidakamizwa egazini kufinyelelwa mayelana amahora ayisithupha.

Ukuxhumana amaprotheni imayelana 99,7%. Ngokuphathelene ukusatshalaliswa ivolumu, khona-ke kusho ukuthi incane (mayelana 0.2 l / kg).

Ngokusho ochwepheshe, tamsulosin lungekho ngaphansi "pass lokuqala" ngokusebenzisa isibindi akheka kancane ukuze metabolites esingasebenzi. Ingxenye enkulu yale ndawo kwaziswa angashintshiwe siyenzeka egazini.

Tamsulosin, kuhlanganise metabolites yayo excreted ikakhulukazi umchamo. Mayelana 9% zomuthi livela ingashintshiwe nge nezinso. Ingxenye-ukuphila we ketshezi kuyinto amahora angu-10.

ubufakazi

Ingabe uyazi ukuthi ngayiphi injongo udokotela ezinqunyiwe izidakamizwa iziguli ezifana "Proflosin"? Analogs ngokwayo, wathi izindlela okudingeka zithathwe kuphela ukwelapha Hyperplasia (ingozi) wendlala indlala, kanye ukwelapha izifo dizuricheskih.

Izimo

Kungaphansi kwaziphi hhayi izimo kungathatha Amaphilisi "Proflosin"? ochwepheshe lezivakashi bathi izidakamizwa akufanele isetshenziswe uma hypersensitivity kuya tamsulosin noma nezinye izinto izindlela, yokwehluleka kwesibindi (ifomu ezinzima), kanye hypotension orthostatic (kuhlanganise umlando).

Ngaphezu kwalokho, i-nomuthi okukhulunywa kufanele kuthathwe ngokuqapha in iziguli nesifo esingamahlalakhona kwezinso futhi lwemithambo hypotension.

Umthamo zomuthi nendlela osebenza ngayo

"Proflosin" - umuthi kwezokuphatha ngomlomo. Ngokuvamile, iqondiswa i nenani capsule lokuqala kanye ngosuku emva ukudla 1st noma kwasemini.

Umuthi kumele wonke kugwinywe (hhayi nganoma iyiphi indlela musa ukuhlafuna), wageza phansi ngamanzi afudumele. Kulokhu, lo capsule akunakwenzeka ukusiqeda noma locezu. Kungenjalo-ke lokhu kungathinta izinga ukukhululwa isithako esebenzayo. Isikhathi izidakamizwa akugcini.

ukweqisa izidakamizwa

Yiziphi ngemiphumela lesiguli kulindeleke uma izidakamizwa "Proflosin" senziwe umthamo omkhulu? Kuze kube manje, amacala ukweqisa izidakamizwa lapho usebenzisa lolu izidakamizwa babonakala. Nokho, ochwepheshe baxwayisa ngokuthi kukhona amathuba ukwehla elibukhali blood pressure kanye okuvela tachycardia. izenzakalo ezinjalo kungadinga amagadango akhethekileko. Ukubuyisela wegazi nokushaya kwenhliziyo kuyehla, isiguli kufanele uthathe evundlile. Hemodialysis kulokhu zingenzeki ngenxa isithako nomuthi has ziyezwana ephezulu Amaprotheni egazi.

Ukuze uvimbele ukumuncwa obengeziwe tamsulosin esiswini ukugeza iyadingeka, futhi ukunikeza isiguli namalahle isebenze noma laxative osmotic.

Ukusebenzisana neminye imithi

Njengoba "Proflosin" yezidakamizwa ithinta edonsa lezinye izidakamizwa ke? Ngokusho kochwepheshe, tamsulosin akusho uxhumane "enalapril" kusho "Atenolol" "Theophylline" futhi "Nifedipine".

Ngekusetjentiswa kanyekanye ne "cimetidine" kukhona ukwanda kancane lokuhlushwa ingxenye esebenzayo olucutshungulwayo izimali e oketshezini olungenambala lwegazi, kodwa "Furosemide" Ngakolunye uhlangothi, ukwehlisa ke. imihlola okunjalo angadingi ukulungisa umthamo nomuthi, ngoba lokuhlushwa yayo lahlala uhla evamile.

Amalungiselelo "Warfarin" futhi "diclofenac" kungaba ngokuphawulekayo ukwandisa izinga excretion of tamsulosin.

ukwelashwa Ngesikhathi tamsulosin nabanye blocker ai-adrenoceptor kungadala ukwehlisa wegazi.

side effects

Senza imiphumela izidakamizwa ecaleni ezifana "Proflosin"? Imiyalelo (imithi efana banikwa ngezansi) uthi lokhu izidakamizwa empeleni umonakala umzimba womuntu.

Cabanga imiphumela emibi izidakamizwa kabanzi:

  • Inhliziyo negazi izitsha: hypotension orthostatic futhi tachycardia.
  • isimiso sezinzwa: isiyezi, yokufikelwa kanye bekhanda.
  • ipheshana wokugaya ukudla: ukuqunjelwa, ukucanuzela kwenhliziyo, isifo sohudo kanye nokuhlanza.
  • System ezalayo: priapism futhi ejaculation sifo.
  • Skin nezicubu ongama iziyaluyalu: ukuqubuka, urticaria, pruritus futhi angioedema.
  • Okunye: ukuthuthukiswa ewumngcingo umfundi syndrome phakathi nokuhlinzwa ngoba cataract, rhinitis futhi asthenia.

Izixwayiso

Yini isiguli phambi nika kunesidingo ukwazisa izidakamizwa yokubika? Ngokusho imiyalelo, umuthi inikezwa kuphela ubulili namandla.

Ngesikhathi izimpawu zokuqala of hypotension orthostatic, isiguli kufanele akhiphe isikhundla ehlezi noma behlezi.

Ngaphambi ukwelashwa kufanele akhiphe khona izifo kanye nezimo ezingaba ukunquma symptomatology efana izimpawu of wendlala Hyperplasia (ingozi).

Ngaphambi ukwelashwa, kanye ngesikhathi kufanele njalo kwenziwe ukuhlolisisa rectal (umunwe).

With ukuthuthukiswa angioedema ukwelashwa kufanele ngokushesha ayisekho. Ukunikeza aphoyintimenti zomuthi is contraindicated.

Lapho ukuhlinzwa elokususa cataract ku ngemuva ukusetshenziswa kwezimali "Proflosin" angagcina ewumngcingo umfundi syndrome. Lokhu kungenzeka kufanele kucatshangelwe ohlinzayo.

Ngesikhathi yokwamukela, ukubika imithi edingekayo ukuze uqaphele ikakhulukazi ngenkathi ushayela, kanye imisebenzi imisebenzi enobungozi okudinga anda okuhlushwa.

Umuthi 'Proflosin ": nozakwabo futhi izindleko imithi

Ingabe uyazi ukuthi kumele ukuthi abantu abaningi abakubheka njengomklamo umuthi? Pharmacy, 30 amaphilisi angathengwa 420-450 ruble Russian. Uma wabelwe Yiqiniso eside yokwelashwa, kwakuzothatha amaphilisi 100. isamba okunjalo zomuthi kubiza ruble mayelana 1,200.

Imiphi imithi ungayithola enye indlela "Proflosin"? kumakhophi are izidakamizwa ezilandelayo: "Tamsulosin", "Bazetu" "Tamsulosin kuthiye ukukhula ',' Fokusin", "hypersimple", "Tulozin", "Glansin", "Taniz-K," "Omnic", "Taniz Heras" "Omsulozin", "Tamsulon-FS", "Revokarin" "hydrochloride tamsulosin" "Sonizin", "Tamzelin" "tamsulosin-Teva".

Le mithi izindlela ezihlukene. Kule ndaba, kufanele ingasetshenziswa kuphela kuma-oda kadokotela.

Uphenyo nomuthi

Yini iziguli elikushoyo ngalokhu imithi, njenge "Proflosin"? Izibuyekezo iziguli akhayo kuphela. Ngokwe-amadoda, abaye wabhekisela capsule, umuthi ngempumelelo ephatha Benign Prostatic Hyperplasia futhi dizuricheskie iziyaluyalu bebonke. Nokho, iziguli eziningi bedidwe izindleko eziphakeme izidakamizwa. Ikhumbula ukuthi kufanele kuthathwe izinyanga eziningana, ukuphathwa eqolo.

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