ImpiloAmalungiselelo

Ama-antibiotic "Glewe": izibuyekezo odokotela

Yini-ke nokuthi ukusebenzisa izidakamizwa "Glewe 500"? Yokusetshenziswa, izilinganiso izici nomuthi wathi ibuye ichazwe. Futhi e mathiriyeli lo sihloko uzothola izimpawu ukuthola le imithi nemikhawulo ngokusetshenziswa kwayo.

Packaging izidakamizwa, yayo ukuma, incazelo, ukwakheka

Ngayiphi ifomu ekhiqizwa izidakamizwa "Glewe?" Izibuyekezo bathi izidakamizwa kufika emashalofini Pharmacy ngesimo amaphilisi. Ziyakwazi ifilimu camera isitini-bomvu, ifomu isiyingi futhi we-lenticular wangakwesokunxele, kanye iphutha umugqa ngakolunye uhlangothi.

Equkethe izidakamizwa "Glewe?" Uphenyo odokotela babike ukuthi imfuyo esemqoka yalolu umuthi levofloxacin. Futhi-ke yakhiwa nezinsizasenzo ezifana crospovidone, microcrystalline cellulose, povidone, isitashi, futhi magnesium stearate.

Ngo ukwakheka amaphilisi equkethe igobolondo: phthalate dibutyl, hypromellose, ama-titanium dioxide, macrogol, udayi obomvu (yensimbi oxide) kanye talcum.

Ngo ukudayiswa izidakamizwa "Glewe" iza ibhamuza amaphakethe, okuyinto zahlanganiswa ngo amakhadibhodi amabhokisi.

Isenzo zomuthi

Siyini "Glewe 500"? Yokusetshenziswa, ukubuyekezwa bathi umenzeli elwa namagciwane bohlanga fluoroquinolone (has a spectrum ezibanzi umsebenzi).

Izingxenye eziyisisekelo lokhu izidakamizwa (levofloxacin) iyakhona ivimbela DNA gyrase (topoisomerase isb 2), futhi topoisomerase 4. Ngaphezu kwalokho, izidakamizwa kanye crosslinking unika supercoiling ye-DNA amakhefu, suppresses zamagama alo, kubangela izinguquko morphological (ezijulile) e ulwelwesi, cell izindonga kanye cytoplasm kwamagciwane.

Izidakamizwa "Glewe", ukubuyekezwa zazo axutshwa, iyasebenza ngokumelene nezilwanyana ezincane eziningi igremu-HIV aerobic.

Izici kinetic

Lapho ukumuncwa lesi sidakamizwa "Glewe?" Imiyalelo, ukubuyekezwa babike ukuthi uma uthatha imithi ye ngomlomo ngokushesha futhi ngokuphelele ugxile kusukela esiswini. Ukudla Ukuthola cishe akunamthelela ukuphelela futhi ngesilinganiso ukumuncwa zomuthi.

I bioavailability ye-ejenti kuyinto 99,5%, kanti lokuhlushwa esiphezulu egazini waphawula ngemva 2 h.

Nathi zemithi plasma amaprotheni cishe 33-40%. It lingena kahle ku izicubu kanye izitho, ikakhulu emaphashini, phlegm, mucosa bronchial, polymorphonuclear leukocyte, izinhlaka uhlelo urogenital futhi macrophage alveolar.

Esikhathini isibindi, ingxenye encane izidakamizwa noma deacetylated oxidized.

Isikhathi isigamu-ukuphila umuthi amahora 6-8. It is lusobala kukho emzimbeni nezinso.

ubufakazi

Lapho ukusebenzisa ejenti antibiotic "Glewe?" Uphenyo odokotela bathi lokhu ejenti liphumelele Izifo ukuvuvukala futhi ezithathelwanayo ezibangelwa amagciwane ebucayi emuthini. Ngakho, imithi kuncike ezinqunyiwe izifo:

  • ENT (kuhlanganise sinusitis acute);
  • izifo (kuyinkimbinkimbi futhi kube lula), izinso kanye ngomgudu womchamo (kuhlanganise prostatitis acute, pyelonephritis uhlobo);
  • ipheshana zokuphefumula, noma kunalokho uqhekeko olukhona ngaphakathi ephansi (kuhlanganise i-pneumonia sinenkonzo yokunakekela iziguli emakhaya kanye ukucinana kwemigudu yokuphefumula acute, uhlobo ezingamahlalakhona);
  • izitho zangasese;
  • komgodi ongaphakathi kwamathumbu (lihambisana ejenti ukuthi isinyathelo izitshalo anaerobic);
  • izicubu zomzimba ezithambile kanye isikhumba (kuhlanganise iqhubeka atheroma, imihuzuko kanye abscesses).

Uvala ukusetshenziswa

Kungaphansi kwaziphi izimo akufanele inikezwe imithi elwa namagciwane "Glewe?" Izibuyekezo usho Izimo ezilandelayo leli thuluzi:

  • ngesikhathi sokukhulelwa;
  • isithuthwane;
  • yobudala ezincane;
  • umonakalo umsipha, okuyinto livelile ngesikhathi azibambile quinolones yokwelapha;
  • ibele;
  • hypersensitivity kuya levofloxacin nezinye fluoroquinolones.

Nge ukuqapha okukhethekile izidakamizwa kubhekwe kufanele sinikezwe abantu abadala kanye (ngenxa awokuthi izinso umsebenzi ukunciphisa), kanye nokuntuleka zikashukela-6-phosphate dehydrogenase.

Tablets "Glewe": yokusetshenziswa

Izibuyekezo babike ukuthi imithi esithathwayo ngomlomo kabili ngosuku. Izibhebhe kufanele kugwinywe iyonke. betel yabo kungavunyelwe (mhlawumbe baphuze eziningi ezanele amanzi).

Umuthi ingagxila ngaphambi kokudla noma phakathi ukudla.

I umthamo we-ejenti kunqunywa kobukhulu kanye nohlobo ukutheleleka, kanye nozwela lwegciwane.

  • Lapho nomuthi iqondiswa sinusitis 500 mg (kanye ngosuku) amasonto amabili.
  • Phakathi exacerbation of ezingamahlalakhona ukucinana kwemigudu yokuphefumula uhlamvu - 250 noma 500 mg (kanye ngosuku) ngeviki.
  • Lapho i-pneumonia CAP - 500 mg (kabili ngelanga) amasonto amabili.
  • Ngo ayinzima pheshana urinary nezifo uhlamvu - 250 mg (kanye ngosuku) izinsuku ezintathu.
  • Prostatitis - 500 mg (kanye ngosuku) inyanga eyodwa.
  • Lapho pheshana urinary nezifo nzima nemvelo (kuhlanganise pyelonephritis) - 250 mg (kanye ngosuku) izinsuku ezingu-10.
  • Lapho elithambile izicubu izifo kanye isikhumba - 250-500 mg (kabili ngelanga) amasonto amabili.
  • Izifo of ngaphakathi komgodi ongaphakathi kwamathumbu - 500 mg (kanye ngosuku) amasonto amabili (lihambisana ejenti elwa namagciwane ayisukumele izitshalo anaerobic).

Lapho kahle umsebenzi sesibindi Ukukhetha okhethekile umthamo liyadingeka, kusukela levofloxacin umzimba hepatic kwenzeka ngezinga elincane.

Ukuze asebekhulile sokuphuzisa umbuso ushintsho ayidingekile, ngaphandle QC ongaphakeme.

Ukwelashwa nale izidakamizwa kumele baqhubeke amahora mayelana 48-78 emva ukuqedwa kanye ukuzinza lokushisa komzimba.

Yeqa yokwamukela nomuthi kufanele kube njengoba fast ngangokunokwenzeka ukuthatha iphilisi. Ngokulandelayo, kudingeka siqhubeke sikhula ngokomoya ukusetshenziswa lwemithi izidakamizwa ebekiwe.

isinyathelo uhlangothi

Yiziphi imithelela uhlamvu omubi umuthi "Glewe 500"? Izibuyekezo ukhombe ukusabela elandelayo:

  • isicanucanu, wehlise blood pressure, ukuhlanza, nciphisa semithambo, uhudo, kahle kungakhuphula izinga likashukela, ukuqunjelwa;
  • arthralgia, ukungakuthandi ukudla, ukuba buthakathaka kwezicubu, ubuhlungu besisu, angaboni kahle futhi ukulalelwa;
  • enterocolitis pseudomembranous, nephritis interstitial, umsebenzi anda transaminases isibindi, rhabdomyolysis;
  • hyperbilirubinemia, ukuwohloka iphunga nokunambitheka kanye ethintekayo ukuzwela, isifo sokusha kwesibindi, tendinitis, dysbacteriosis;
  • myalgia, tachycardia, ukwehluleka oyingozi so-renal, urticaria, fibrillation atrial;
  • ikhanda, hypercreatininemia, isiyezi, anaemia hemolytic, ubuthakathaka, agranulocytosis;
  • somnolence, isikhumba kanye mucosal edema, ukuqwasha, ukushaqeka anaphylactic, liqhaqhazela, vasculitis, ukukhathazeka neutropenia, paresthesias;
  • hypersensitivity pneumonitis, ukwesaba, ukubindwa, ukuhhema, eziya ziba zimbi ka porphyria, ukudideka, pancytopenia;
  • ukucindezeleka, ukuntuleka kwegazi emzimbeni, ukunyakaza neziyaluyalu, imfiva ophikelelayo, ukuquleka, umsipha ukudabuka;
  • leukopenia, ukulunywa futhi isikhumba ngamanzi, asthenia, erythema exudative abulalayo, eosinophilia;
  • necrolysis epidermal anobuthi, bronchospasm, ukuthuthukiswa superinfection, ukopha, photosensitivity.

Analogs kanye nezindleko

Intengo leli thuluzi ruble mayelana 170-250. Kwezinye izimo, lokhu izidakamizwa esikhundleni izidakamizwa ezifana "Levolet", "sol", "Toksof", "Lebel", "Levofloxacin", "Levobaks", "Levofloks", "Levobakt", "Levotor", "Levokilz" "Levostad", "LeVox," "Levomak", "Levoksimed".

Ama-antibiotic "Glewe": Izibuyekezo iziguli nodokotela

Umthengi Izibuyekezo mayelana izidakamizwa "Glewe" elixutshwe. Abakwazi ahlukaniswe abe amaqembu 2: omunye ithonya ujabule izidakamizwa, ngoba kuyakusiza ukuba sibhekane ngokuphumelelayo nezifo ezithathelwanayo nge sakugcina izigameko ezingezinhle ezavela kanye nezinye - uthe izidakamizwa ayizwakali.

Ngokuqondene odokotela, umbono wabo ukuthi izidakamizwa "Glewe" kuyinto-antibiotic eqinile ukuthi ingase ikhishwe kuphela ngemva kokukhuluma nodokotela. By the way, ochwepheshe abaningi kubhekwe ngokuhlanganyela imithi Kunconywa ukuthatha probiotics, ukuze onakalise microflora emathunjini.

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