ImpiloAmalungiselelo

"Captopril". Yokusetshenziswa

"Captopril» (captopril) - umuthi okuqondene iqembu angiotensin ukuguqulela enzyme inhibitor (ACE inhibitor). Esikhathini ngamazwe ngezigaba uhlelo izidakamizwa "Captopril" ikhodi yokubhalisa C09AA01. Engama synthetic chemicals ukulungiselela "Captopril" kuhloswe ukuba kunciphise umfutho wegazi ngokunciphisa hormone kumiswa oligopeptide (eyatholakala kusukela angiotensin mina angiotensin II), okuholela ukwehla ekukhiqizeni i-adrenal cortex i-hormone mineralokortikosteroidnogo - aldosterone.

Kukhona amagama akho okuhweba eziningana abakhiqizi ezahlukene ukukhiqiza "Captopril" ngaphansi kwazo. Ukusetshenziswa kwe-brand ngamunye Guide echaza umumo nokukhululwa umthamo (ngokuvamile izibhebhe 6,25 mg, 12.5 mg, 25 mg, 50 mg, 100 mg). "Sesifufula Okwemithi" umkhiqizi - "Angiopril 25" amaphilisi. "Vokhard Limited" - "acetyl". ezithaka imithi prdktsii enkulu kunazo zonke emhlabeni "Bristol-Myers Squibb" igcwalisa izibhebhe emakethe "Capoten". Inkampani Russian "Akrikhin" ukhiqiza "Capoten". Tablets ngaphansi "Captopril" lokuhweba ekhiqizwa amafemu eziningana: "Elfa" (Russia), "hexane" (eJalimane), "Krka" (Slovenia) "Promed Exports" (Russia), "Rompharm" (Russia). Inkampani American "Ai-CN Okwemithi" ukhiqiza "Katopil" amaphilisi-mbumbulu. Oholela Inkampani ekhiqiza imithi EGrisi "Medokemi" - "Rilkapton". Hungarian ezithaka imithi ifektri "Aegis" - amaphilisi Tenziomin. inkampani yaseKhupro "Remedika-Minneks" - "Epsitron".

Odokotela ukunquma "captopril" monotherapy ngokwanda ziphikelele komfutho wegazi (hypertension). Umuthi esetshenziswa ekwelashweni amafomu njalo congestive ukuhluleka kwenhliziyo, lapho (ngemva infarction), ngakwesokunxele umsebenzi ventricular. It ezinqunyiwe ekwelapheni nephropathy sikashukela, okwenzeka ngokumelene isizinda sikashukela uhlobo lokuqala. umphumela Lokulingene hypotensive, nezinye ACE inhibitor inikeza ukwehla okuphawulekayo wegazi. Ezimweni eziningi isigamu umthamo esiphezulu umthamo ibekezelelwe zomuthi kwanele. Uma kuqhathaniswa neminye imithi, njenge hydrochlorothiazide, kancane side effects, inikeza "Captopril". Yokusetshenziswa uchaza umthamo wakhe ngqo.

Ukuthuthukisa hypotensive "Captopril" umphumela sisetshenziswa ndawonye nezinye izidakamizwa: isisu (isisu - hydrochlorothiazide), noma -calcium channel blocker (calcium abamelene nge evelele vasodilator isenzo - verapomil, nifedipine nabanye). Kuphela ngesisekelo inhlolovo, futhi esekelwe yobudala kanye isimo jikelele zomzimba, udokotela (lihambisana namanye izidakamizwa noma monotherapy Yiqiniso) inikeze "Captopril". Yokusetshenziswa zomuthi kufanele wafunda yisiguli, kodwa ukushintsha Isikali yabo ukukhansela inkambo udokotela, noma akufanele self-medicate. Uma kungenjalo, kungaholela emiphumeleni engathí sina ezimbi.

Udokotela ubeka umuntu izidakamizwa nokushintsha kokudla nokufakwa lwemithi. Ngokuvamile ihora ngaphambi kokudla Kunconywa ukuthatha "Captopril". Ukusebenzisa izidakamizwa kufanele kube njalo, ngesinye futhi ngesikhathi esifanayo. Lapho umfutho wegazi ophakeme "Captopril" ngokuvamile eyabelwe 25 mg (kabili ngelanga). Ngemva kwalokho umthamo kungase kukhule kancane kancane kuze kube nomphumela ofiselekayo abayifunayo. Ukuze ngokulinganisela blood pressure yakhe senyuselwa 50 mg (kabili ngelanga), futhi ifomu ezinzima zalesi sifo izidakamizwa kungenzeka kuze kube kathathu ngosuku ngo-50 mg. Kulokhu, lo umthamo wansuku zonke kumele singeqi 150 mg. Zonke yalezi zinguquko kumele kwenziwe Isikali udokotela. Okungalapheki inhliziyo ukwehluleka kanye uswidi "captopril" , Isikali ukuqala 6,25 mg izikhathi ezintathu ngosuku. Khona-ke, lokhu umthamo kungenziwa kancane kancane, kodwa hhayi ningi than suku 150 mg. ezigulini esezikhulile kanye neziguli nge kahle umsebenzi kwezinso acophelele kakhudlwana lapho eshayela esimisiwe 'Captopril ". Yokusetshenziswa zomuthi iqukethe ulwazi Izimo kanye nezinkinga kungenzeka ukuthi isiguli akufanele sikhohlwe sihlale njalo siqaphele isimo sabo. Uma kudingeka, "Captopril" kuthathwe kanye isisu thiazide uchungechunge (hydrochlorothiazide, chlorothiazide), noma iluphu isisu (isib furasemid).

Ulwazi oluqukethwe kulesi sihloko akusho ukuthi akufanele kusetshenziswe lodokotela.

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