ImpiloAmalungiselelo

"Driptan": ukubuyekezwa. "Driptan": yokusetshenziswa, intengo

Wonke umuntu phezu esaphila kungase uhlangabezana nezinkinga ezihlukahlukene obuseduze, okuyinto angifuni ukukhuluma, futhi uma kunesidingo, ngakho kuphela, bazethula. Enye inkinga enjalo kuyinto incontinence urinary. Kungenzeka njengoba izingane ezincane kanye omdala. Incontinence kungenziwa ebonakaliswa yezifo ngomgudu womchamo abese e kwempilo yengqondo. Uma ukuchama njalo futhi bengaphazamisekile, kodwa kukhona incontinence, lokhu kuwubufakazi bokuthi kwezinso zokukhula esinyeni neziteshi urinary. Endabeni incontinence, akunandaba yini isizathu sale nkinga, odokotela bavame linqume izidakamizwa "Driptan" Izibuyekezo nesineke abonisa ukuthi le sidakamizwa sisiza ukuqeda lezi zenzakalo edabukisayo. "Driptan" buyisidakamizwa ukuthi kunciphisa bushelelezi imisipha ithoni kwesinye futhi ngomgudu womchamo.

Sakhiwo Ukwakheka

The main isithako yalesi izidakamizwa izenzo oxybutynin hydrochloride. Futhi kule "Driptana" kuhlanganisa excipients ezihlukahlukene ezifana ne-lactose, microcrystalline cellulose ne-calcium stearate.

Umuthi itholakala ngendlela amaphilisi isiyingi kokuba umbala omhlophe. Biconvex ifomu ithebhulethi, ngakolunye uhlangothi kukhona ingozi kakhulu kulolu phiko.

Kokunye ibhamuza kuyinto amaphilisi 30. Umuthi itholakala ngaphatha ibhokisi elinezincwadi, okungase elilodwa noma amabili amabhamuza.

imiphumela kwemithi

Medicine "Driptan" libhekisela eqenjini kwemisipha relaxants. Umuthi has a action antispasmodic futhi anticholinergic m-myotropic oqondile. Kusho ikhuthaza ukuphumula we detrusor nokunyusa umthamo esinyeni. Ngaphezu kwalokho, ngenxa yalokhu izidakamizwa encishisiwe ukuvama Kufinyeta we detrusor futhi ayenele by nesifiso sokufuna ukuchamela.

Pharmacokinetics

Ngemva contact zomuthi emzimbeni womuntu kufinyelelwa emva kwemizuzu 45 C max. Umthamo umuthi wakhona okuhlushwa.

izinkomba Sebenzisa

Umuthi 'Driptan "ingasetshenziswa yibo bobabili abadala kanye nezingane. Leli thuluzi wenziwa engabelwe abadala endabeni detrusor ukuntengantenga nemisebenzi incontinence. Nokuntengantenga kwesinye kanye wokuphuthuma uma Uphinde abhekwe izinkomba ukusetshenziswa "Driptana". Futhi, lolu izidakamizwa isetshenziswa idiopathic esinyeni overactive futhi ukuchama kaningi. Ngokuvamile i-ejenti isetshenziswa ukulawula hyperactivity kwesinye, okungase kwenzeke phakathi cystitis, futhi ngemva kokuhlinzwa ku esinyeni noma wendlala.

Bangase babe 'Driptan "izingane incontinence noma ukuchama kaningi. I izinkomba ukusetshenziswa kwalesi izidakamizwa ezinganeni kungenza njengesithiyo i esinyeni umsebenzi engazinzile ngenxa ukungasebenzi neurogenic. enuresis Nocturnal futhi inkomba kokuthola ithebhulethi idatha. Abantwana kwenzeka adiopaticheskaya ukungasebenzi, okuholela ukhombe "Driptan". Uphenyo odokotela wabonisa ukuthi isidakamizwa kahle kubekezelelwe izingane, okuyinto isheshisa ekusimameni.

Izimo

I contraindication umzimba sokuqala hypersensitivity imithi izidakamizwa esebenzayo noma ama-ejenti asizayo main. Futhi, izidakamizwa is contraindicated ebantwaneni ngaphansi kweminyaka engu-5. Awukwazi ukusebenzisa izidakamizwa ngesikhathi enomkhuhlane, + futhi ngaso okushisa ephakeme. Umuthi akuyona efiselekayo ukusebenzisa ngenkathi bekhulelwe nangenkathi bencelisa. Medicine "Driptan" kwenqatshelwe ukuyisebenzisa ngoba ezinzima izilonda emathunjini bese pheshana urinary isimiso.

Ngaphezu kwalokho, i-ejenti akuthathi yezifo ezifana myasthenia gravis, ewumngcingo-engela ukufiphala ipayipi lokukhipha indle, megacolon anobuthi, ileostomy, ezofagelnaya ukungasebenzi. Izimo ukusetshenziswa kwezidakamizwa futhi organic, ileus obusebenzayo noma kofé uhlangothi, futhi atony emathunjini bese stenosis pyloric.

"Driptan": Isicelo (imithetho eyisisekelo)

Lesi sidakamizwa esithathwayo ngomlomo ngaphakathi. Adult kufanele ukuthatha imithi 2-3 izikhathi 1 ithebhulethi suku. Ithebhulethi ingahlukaniswa ngesigamu ngoba isicelo kulula. Umthamo esiphezulu oxybutynin hydrochloride ngelanga 20 mg.

ezigulini esezikhulile kufanele athathe izidakamizwa lapho kugamanxa iphilisi 2 izikhathi ngosuku. Uma kudingekile, futhi ngaphansi kokuqondisa okuqinile udokotela, ungathatha wonke tablet futhi izikhathi 2.

"Driptan" izingane letimisiwe ithebhulethi ngosuku, ukukucaza kube 2 imithamo. Futhi ucabange yokwamukela 2 amaphilisi ngelanga, kodwa ngaphansi kokuqondisa kukadokotela.

isicinganani

"Driptan 'linenani elikhulu amathuba okuba nemiphumela engemihle.

  • Ngokuphathelene ipheshana wokugaya ukudla: bangezwa isicanucanu, nomlomo owomile, ukuhlanza, kabi noma ubuhlungu esiswini, uhudo noma ukuqunjelwa.
  • CNS: kungaba isiyezi, ukozela, nesimo sokuquleka noma ikhanda. Iphinde zingase zibe zimbi iphango. Ngaphezu kwalokho, ukusangana kungenzeka, ukudideka, ukuyaluza, amaphupho amabi, uhlanyiswa nokukhathazeka disorientation.
  • Isihlobo emehlweni: zingavela angaboni kahle bese we conjunctiva, iso ingcindezi wande, futhi izingane zesikole kuthiwa osuke usuvulekile (njengoba kuboniswa exhunywe izidakamizwa "Driptan" yokusetshenziswa). Izibuyekezo luye lwabonisa ukuthi imiphumela emibi ezingavamile, ngenkathi kancane obonakalayo.
  • Ngokuphathelene izinso kanye urinary iziteshi kungenzeka dysuria kanye nokugcinwa umchamo.
  • Ngokuphathelene inhliziyo: mhlawumbe ibonakalisa arrhythmias inhliziyo, ukufikelwa ukushisa kanye tachycardia.
  • Futhi kungenzeka isikhumba ukuphendula. Ngokwesibonelo, amawala, ezomile, edema angioneurotic noma isifuba.

Ukuze ugweme side effects, kumele uthathe ngokucophelela izindlela "Driptan". Izibuyekezo baye babonisa ukuthi isidakamizwa kahle ikubekezelele izingane kanye nabantu abadala, uma wamukelwe ngendlela esiyalwe ngayo.

ukweqisa izidakamizwa

Umhlahlandlela uxwayisa ngokuthi ukweqisa izidakamizwa yalesi izidakamizwa kungaba. Uma kwenzeka yokudlula umthamo izidakamizwa kungabonakala nasemkhakheni izimpawu ezifana ukusangana, Ukudlikizela, liqhaqhazela, ukukhathazeka, delirium. Kungase kubangele ukwethuka, imfiva, ukuhlanza, isicanucanu. Kungase futhi wehlise blood pressure, cishe kubonisa tachycardia nokuvaleka kwemigudu yokuphefumula. Ezimweni ezimbi kakhulu kakhulu kungenzeka ukukhubazeka, futhi equlekile.

Ukuze balahle izimpawu ngokweqile, kubalulekile ukuba iphume esiswini futhi uthathe carbon isebenze, ingabagulisa ukuhlanza eyayenziwe noma usebenzise nosawoti laxatives. Uma kudingekile, udinga basekelwe ukuphefumula. Ukuze ususe izimpawu ubuthi anticholinergic, blocker cholinesterase kumele kusetshenziswe. Lokhu okwashiwo yilo mlobi liphinyiselwe inexhala noma ukucasuka, faka 10 mg diazepam. Uma tachycardia kubonakala - e / propranolol.

izidakamizwa ekuhlanganyeleni

Uma uthatha le imithi kanye "lisuride" singenzeka ukuphazamiseka ukwazi. Kufanele kusetshenziswe ngokuqapha kulesi izidakamizwa kanye namanye amanxusa anticholinergic, hhayi potentiate imiphumela anticholinergic.

Futhi "Driptan" ayikwazi ukusetshenziswa ngokuhlanganyela butyrophenones, phenothiazines, tricyclic antidepressant, amantidine futhi levodopa. Ngemva kokuthola lezi "Driptana" kwenzeka esiswini motility ukunciphisa, ngenxa okungase ziwohloka absorbitsiya nezinye izidakamizwa. Hlanganisa utshwala nale izidakamizwa is hhayi Kunconywa.

"Driptan" ngesikhathi sokukhulelwa

Phakathi nenkathi yokukhulelwa, le edonsa izidakamizwa kungenzeka, kodwa kuphela uma kukhona phezu izinkomba esiqinile. Kungcono ukuthatha izidakamizwa ngaphansi kweso lwezokwelapha. Uma ukwamukela kusho kuyadingeka esikhathini lactation kufanele kube isikhathi ukuyeka ibele.

imiyalelo Special

Ngakho umuntu kufanele aqaphe ukuthatha izidakamizwa iziguli esingamahlalakhona nephritic futhi hepatic. Iziguli-hyperthyroidism, futhi ukumelwa inhliziyo, kanye nalabo abaphethwe arrhythmia, noma umfutho wegazi ophakeme, futhi kumelwe siqaphele ukuba afeze amaphilisi.

I inani lentengo lomuthi

Kuthathwa ukuba izidakamizwa kuqhathaniswa eqolo "Driptan". Intengo ke Pharmacy ezahlukene kuhluka ruble 1,000 ukuze 1,500 iphakethe ngalinye, lapho 30 zithutha.

I-ejenti

Umuthi kufanele igcinwe kude nezingane. okushisa Isitoreji kumele singeqi degrees 28. Shelf-ukuphila umuthi izinyanga 36. Okunikelwa enemithi.

"Driptan": nozakwabo

Ngenxa yokuthi lo muthi ikhishwe kuphela kadokotela we udokotela, kaningi Pharmacy ukubuza esikhundleni. Kufanele uthintane usokhemisi umtshele ukuthi ngasizathu simbe, wathenga izidakamizwa, njengoba lisho amaqembu imithi emibili. Ithathwe ayephuli ukuchama - iqembu lokuqala lapho "Driptan". Analogue kuleli cala - kuyinto "Vero Pigeum" "Capsicum-plus", "Aktipol". Iqembu lesibili - izidakamizwa ukuthi ebekiwe bedwetting. Leli qembu kuhlanganisa "Apo-Famotidine."

Izibuyekezo sokulungiselela

Baningi abadala nezingane ngisho nasebekhulile omuhle kuphela ngalokhu nokulungiselela. Umama, okwadingeka ukuba anikeze amaphilisi izingane zabo nabo bayakholelwa ukuthi leli izidakamizwa kuye kwaba nomphumela omuhle futhi kahle ikubekezelele seziguli ezisencane.

Kukhona banombono ongemuhle mayelana izidakamizwa "Driptan". Uphenyo abanye abadala baye babonisa ukuthi izidakamizwa akuzange kusize ukuqeda lesi sifo, futhi lapho ethatha wabonakaliswa ubuhlungu besisu, okuyinto wanyamalala ngemuva ukuqedwa zomuthi. Kodwa ukuze izidakamizwa enikeziwe isenzo edingekayo, kufanele kuthathwe kuphela ngaphansi kweso lwezokwelapha.

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