ImpiloAmalungiselelo

"Sulphate Gentamicin": yokusetshenziswa, analogs kanye nokubuyekeza

izinqubo eziningi ezithathelwanayo kanye ukuvuvukala emzimbeni ngeke akwenze ngaphandle ukusetshenziswa kwemithi elwa namagciwane. Iqembu zalezi zimali obulala amagciwane ayingozi futhi Amagciwane. Omunye namagciwane eyaziwayo "Gentamicin sulfate." He kubhekwa ama-antibiotic nge spectrum ezibanzi izicelo futhi lusetshenziselwa ukwelapha abantu kanye nezilwane.

Ukuma kanye nendlela okwakheke ngayo izidakamizwa

izindlela Iyatholakala ngesimo 4% isixazululo imijovo iso amaconsi. The main izidakamizwa ketshezi Ukwakheka kuyinto sulfate gentamicin umthamo 4 mg ngemililitha ngayinye. Lihlobene aminoglycoside iqembu futhi ubhekwa ezibanzi-spectrum antibiotic.

Umuthi has isinyathelo eqeda ukuvuvukala kanye amagciwane. It has a umsebenzi omkhulu ngokumelene anaerobic amagciwane igramu-negative futhi cocci igremu-HIV. Ngemva kokuphathwa esicutshini zomuthi ngokushesha ugxile. Umthelela esiphezulu kufinyelelwa ngemva kwamahora ambalwa umuntu umjovo. Cishe asisho abophe ukuze Amaprotheni egazi. Okusatshalalisiwe-antibiotic oketshezini extracellular yazo zonke kwezitho izinhlelo. Umuthi akuyona akheka futhi ngokuyinhloko excreted ngu izinso, kancane - ne Bile. It uvame ukuba adabule esinomhlapho isithiyo ekwakhiweni "Gentamicin sulfate." Ukusetshenziswa side effects - konke lokhu kufanele uhlole ngaphambi uhlela ukwelashwa.

ubufakazi

Umuthi kuboniswa ngenxa yezinqubo ezithathelwanayo kanye ukuvuvukala emzimbeni, okuyinto zibangelwa nezilwanyana ezincane ekuthonyweni antibiotic. Ukuze abaphathi parenteral :

  • cystitis;
  • cholecystitis acute;
  • ubovu izilonda zesikhumba;
  • ukusha idigri obuhlukahlukene;
  • pyelonephritis;
  • cystitis;
  • izifo ngisho namalungu amathambo i nature esithathelanayo;
  • sepsis;
  • peritonitis;
  • i-pneumonia.

Lapho ihlelwe ngokulandelana kwezihloko isicelo:

  • imihuzuko;
  • folliculitis;
  • dermatitis seborrheic;
  • ukusha onegciwane;
  • ebusweni nilimaza of omsakazo ezihlukahlukene;
  • sycosis.

Ukuze ukwazi ukufaka isicelo endaweni:

  • blepharitis;
  • blepharoconjunctivitis;
  • dacryocystitis;
  • konyuntivit;
  • keratitis.

wasebenzisa "Gentamycin sulphate" Kulezi pathologies. Yokusetshenziswa kukhona phakathi ekhemisi nge iphakethe imithi.

Izimo:

  • hypersensitivity nemithi;
  • isibindi ezinzima futhi ukwehluleka kwezinso;
  • kokunikezwa kwe-nerve sokuzwa;
  • yokuzala;
  • ibele.

Futhi ayizange inikezwe antibiotic "Gentamycin sulphate" e ampoules e uremia.

Isikali

Linqume izidakamizwa isiguli ngayinye. Umthamo incike ngobucayi inqubo hypersensitivity i-ejenti. Kwelinye ingxenye iqondiswa kusuka 1 kuya 1.7 mg ngayinye esisindo kg. Umuthi iqondiswa ngemithambo yegazi noma intramuscularly. Umuthi isetshenziswa izikhathi ezimbili kuya kwamane ngosuku. Isikali Maximum ngosuku akumele seqe 5 mg. Inkambo yokwelashwa singemaviki lange 1.5.

Izingane emva kweminyaka emibili kwezidakamizwa iqondiswa izikhathi eziningana ngosuku e isamba 1 mg amakhilogramu esisindo ngayinye. Eyenzelwe izingane ezineminyaka engu kuze kube inyanga eyodwa hhayi umthamo nsuku zonke kungaba ezingaphezu kuka 2-5 angu amakhilogramu esisindo ngayinye. I-antibiotic iqondiswa izikhathi eziningana ngosuku.

Ukuze baqonde izinto ezenzekayo amathonsi ocular econsa 1 iconsi njalo ngemva kwamahora amabili. Ukuze zangaphandle ukusetshenziswa ejenti iqondiswa kuze kube kathathu ngosuku. Abantu ne kahle izinso umsebenzi, kuye lwasemtholampilo isithombe ukulungiswa wenziwe ukulungiswa "Gentamicin sulfate." Eye amaconsi bangcwatshwe ngqo ngaphakathi komgodlana conjunctival kwamehlo lesiguli.

Ukuxhumana nezinye izidakamizwa

Akunconyelwe co-ukuphatha ne izidakamizwa ezilandelayo:

  • "Vancomycin";
  • "Cephalosporin";
  • "Ethacrynic acid";
  • "Indomethacin";
  • kusho izinzwa;
  • analgesics;
  • iluphu isisu.

Ngaphambi ukwelashwa ukuhlela, kumele uhlole ngokucophelela nokuxhumana neminye imithi futhi imithi elwa namagciwane "Gentamicin sulfate."

Ngazishaya indiva izincomo kungaholela ukuthuthukiswa okulandelayo side effects:

  • isicanucanu;
  • ukuhlanza;
  • bilirubin zandiswe igazi;
  • anaemia;
  • thrombocytopenia;
  • wegazi;
  • migraine;
  • isiyezi;
  • proteinuria;
  • iziyaluyalu apharathasi vestibular.

Iphinde bangase baxabane nomzimba "Gentamicin sulfate." Amaconsi ikhambi futhi ezimweni ezingavamile kungabangela edema angioneurotic noma ukushaqeka anaphylactic, ezithinta eziyingozi. Ngo ukusetshenziswa lo muthi ezidingekayo ukuqapha umsebenzi izinso, ama-apharathasi sokuzwa kanye vestibular.

"Sulfate Gentamicin" - i-antibiotic ukuze izilwane

Izilwane ezifuywayo nabo basengozini yokugula ukuze kwegciwane. Ukuze ekwelapheni abagulayo iqembu isilwane ekhethekile kwamaphilisi esetshenziswa. "Gentamicin sulfate" libhekisela izidakamizwa ezinjalo. It kungokwalabo iqembu aminoglycosides futhi inhlanganisela gentamicin C1, C2 futhi C1a. Ukwakheka izidakamizwa kuhlanganisa gentamicin 40 no-50 mg kwelinye ngemililitha solution. Kusho agcinwe ezingeni lokushisa hhayi ngaphezu kuka-25 degrees, futhi endaweni eyomile indawo kude nezingane. kweminyaka emibili - izidakamizwa eshalofini yokuphila "Gentamicin sulfate." Yokusetshenziswa izilwane ukukhuluma ngokuningiliziwe mayelana izinkomba kanye umthamo we izidakamizwa.

umphumela

Umuthi has a spectrum ezibanzi imiphumela, futhi umsebenzi ngokumelene igremu-HIV futhi igremu-negative nezilwanyana ezincane. Ngemva kokuphathwa zomuthi isikhathi esifushane lapho ingena phakathi zonke izinhlaka futhi izinhlelo. Ngemva kwehora elilodwa, it is waphawula umsebenzi esiphezulu futhi kuthathe amahora angu-8. Bhala ikakhulukazi umchamo, futhi lokuhlala elincane indle besikhumba saleso silwane.

Umuthi kuboniswa ukwelapha ezifuywayo e pathologies isisu, amathumbu, peritonitis, meningitis, pyelonephritis kanye nezinye izifo. Umuthi iqondiswa kabili nsuku zonke at esingaba amahora 10. Futhi iqondiswa ngomlomo kusho "Gentamycin sulphate" isilwane.

Isikali

Ukuze ekwelapheni amahhashi-antibiotic iqondiswa intramuscularly at umthamo 2.5 mg ngayinye isisindo amakhilogramu umzimba. Ubude besikhathi sokwelashwa imayelana 3 izinsuku ezingu-5. Izinkomo injected umthamo izinga 3 mg amakhilogramu esisindo ngayinye izinsuku 5. Futhi, izidakamizwa ingasatshenziswa ngomlomo ngesikhathi umthamo 8 mg amakhilogramu esisindo ngayinye.

isixazululo Izingulube ukuthi injected intramuscularly ngesilinganiso 4 mg ngayinye isisindo 1 kg. Isikhathi yokwelapha kumele singeqi izinsuku ezintathu. Ngemlomo izidakamizwa isetshenziswa ngesikhathi umthamo 4 mg amakhilogramu esisindo ngayinye izinsuku 5. Izinja namakati ujove esicutshini 2.5 mg isixazululo ngasinye kg esisindo. Ukwelashwa kungathatha izinsuku eziyisikhombisa.

Lapho ebonisa indlela lo izidakamizwa ngaphakathi is hhayi ugxile esiswini kodwa amahora kuphela ngemva kuka-12 emathunjini. "Gentamicin sulfate" kungenziwa kuphela iqondiswa intramuscularly-antibiotic wezilwane. Imiyalo isilwane uchaza izindlela kwezidakamizwa abaphathi.

Izixwayiso

It kungavunyelwe ukusebenzisa ama-antibiotic namanye amaqembu izindlela nephrotic, ikakhulukazi zokugula we kwezinso futhi ubuthulu. Ekuhlatshweni kwezilwane kuvunyelwe ngemva kwamasonto amathathu kuphela umthamo wokugcina izidakamizwa. Ithuluzi engathathi isinyathelo phezu aphansi isikhunta, amagciwane kanye anaerobic amagciwane. Kuphela uchwepheshe wezilwane kungaba kahle ukubala umthamo imithi "Gentamicin sulfate 4%" futhi baphathe isilwane sakho.

Izidakamizwa "Gentamicin"

Umuthi kungokwalabo-antibiotic we aminoglycoside, iziphi kabanzi esetshenziselwa ukwelapha izifo eziningi. Ithuluzi inikeza imiphumela elandelayo emzimbeni:

  • amagciwane;
  • anti-inflammatory;
  • It has umsebenzi omkhulu ngokumelene amagciwane Gram-HIV futhi Gram-HIV.

Umuthi itholakala ifomu isixazululo. Ngemva kokuphathwa esicutshini zomuthi ngokushesha angena ezicutshini zawo wonke umzimba. bioavailability Iningi waphawula ngemva isigamu sehora. Isigamu kusho emva 3 chasa excreted ku umchamo. Kweqa yi-placenta, ngakho-ke, is hhayi Kunconywa ngesikhathi sokukhulelwa, lesi sidakamizwa "Gentamicin" futhi okuphikisana nalo "Gentamicin sulfate." Yokusetshenziswa zalezi zimali inikeza ukwaziswa okuwusizo futhi incazelo kwama-antibiotic.

Izinkomba kanye contraindications

Ukwelashwa kwezifo ezithathelwanayo kanye ukuvuvukala ezibangwa ingxenye zamanje nokuzwela izilokazane ezincane kungase kwenziwe usebenzisa "Gentamycin" lisho ukuthini. Ukulungiswa isetshenziselwa isicelo parenteral, yangaphandle futhi lendawo.

Izimo:

  • Hypersensitivity ukuze aminoglycoside iqembu;
  • yokuzala;
  • lactation;
  • degree okunzima ukwehluleka kwezinso;

Ngaphambi kokuqala inqubo ukwelashwa kufanele uhlole ngokucophelela zonke contraindications nokusetshenziswa kwamaphilisi "Gentamicin" futhi "Gentamicin sulfate."

Isikali

Umuthi inikezwa ngamunye, umthamo incike ngobucayi isifo. Ukuze abaphathi esicutshini noma emthanjeni kusho ibalwa umthamo 1 kuya 1.7 mg amakhilogramu esisindo ngamunye kanye. Ebusuku izidakamizwa iqondiswa izikhathi ezimbili noma ezintathu. Umkhawulo engayitholi nsuku umuntu omdala kumele singeqi 5 mg / kg, futhi izingane - 3 mg ngayinye isisindo amakhilogramu umzimba. Umuthi iqondiswa izinsuku ezingu-7. Eye amaconsi asetshenziswa kathathu ngosuku nokugxilisa eyodwa consi iso abathintekayo ngokushesha. Ihlelwe ngokulandelana kwezihloko isicelo imithi elwa namagciwane kane ngosuku. Ngo ezinzima isifo sezinso ikhambi inikezwa ngokuvumelana isithombe sokucindezeleka, umthamo kungase kushintshwe. Ezinganeni yangosuku incike yobudala kanye nesimo umzimba.

izidakamizwa ekuhlanganyeleni

Kusho "Gentamicin is" hhayi Kunconywa ukuba isetshenziswe lihambisana izidakamizwa ezilandelayo:

  • "Vancomycin";
  • "Cephalosporin";
  • "Ethacrynic acid";
  • "Indomethacin";
  • analgesics;
  • Imithi ye-izinzwa;
  • isisu.

Have ukwakheka efanayo futhi izinkomba ngokusetshenziswa umuthi "Gentamycin" isixazululo kanye "Gentamicin sulfate 4%." Zombili imikhiqizo abe izakhiwo okusezingeni eliphezulu amagciwane anti-inflammatory.

Izidakamizwa "Gentamicin-Verein"

Ucatsanisa aminoglycoside izidakamizwa futhi sisetshenziswa kabanzi ekwelapheni izitho eziningi izinhlelo. Ingabe umsebenzi lakhuphuka lafika ku-Gram-HIV futhi igremu-negative anaerobic amagciwane. It kunomphumela amagciwane. Ngemva ukwethulwa-antibiotic esicutshini futhi emthanjeni angena zonke kwezitho nezicubu zomzimba.

imizuzu engu-40 ngemva umjovo izidakamizwa ifinyelela umsebenzi esiphezulu, okuyinto kuthathe amahora 12. Ithuluzi akuyona akheka futhi excreted ku umchamo. It has ikhono ukungena ngokusebenzisa isithiyo esinomhlapho.

Izinkomba kanye contraindications

Umuthi esetshenziselwa ukusetshenziswa parenteral, lendawo futhi baqonde izinto ezenzekayo ekwelapheni izifo ezithathelwanayo neziyaluyalu ukuvuvukala.

Izimo:

  • ukhulelwe;
  • ibele;
  • ukwehluleka kwezinso nesibindi;
  • hypersensitivity;
  • neuritis we emsipheni sokuzwa.

Isikali "Gentamicin-Verein" izidakamizwa

Kubantu abadala, umuthi injected isamba ezingekho ngaphezu 5 mg ngayinye esisindo amakhilogramu ngosuku. Ngesinye isikhathi, umthamo kuyinto kusuka 1 kuya 1.7 mg ngayinye 1 kg isisindo nesineke. Inkambo yokwelashwa incike kobukhulu inqubo futhi ivela izinsuku ezingu-7 kuya kwezingu-10. Umuthi itholakala izikhathi ezimbili noma ezintathu ngosuku

Ezinganeni, umthamo 3 mg amakhilogramu ekuphathweni esisindo ngamunye. Umuthi waqala kabili ngosuku. Iziguli esingamahlalakhona kwezinso, umthamo we antibiotic njalo kushintshwe futhi kuncike izinkomba zokwelapha.

Eye amaconsi asetshenziswa njalo ngemva kwamahora 4, futhi wangcwatshwa ethintekile iso iconsi. I-ejenti zangaphandle inikezwa kathathu noma kane ngosuku.

Imiphumela engemihle engase ibe:

  • isicanucanu;
  • ukuhlanza;
  • anda bilirubin;
  • anaemia;
  • leukopenia;
  • ukozela;
  • migraine;
  • iziyaluyalu apharathasi vestibular;
  • ubuthulu;
  • komzimba, kuze angioedema.

Okufanayo kahle emzimbeni imithi kunganqotshwa eziyoncibilika 'Gentamicin sulfate 4% "ngesikhathi ekwelapheni izinqubo ezithathelwanayo kanye ukuvuvukala emzimbeni.

Uphenyo gentamicin amalungiselelo sulfate ezisekelwe

Imithi azisebenzi imithi elwa namagciwane of isizukulwane esisha, kodwa okuhle ngokwanele esikhathini sethu isetshenziselwa ukwelapha izifo amagciwane abe nenkani. Ngakho-ke, isethi imikhiqizo okwethulwa emakethe weenhlahla, okuhlanganisa gentamicin. Akukhona izixazululo komjovo kuphela, kodwa futhi okhilimu yokugcoba, ngeso lehla. Umuthi sithinta ukwaziswa kwezakhi zofuzo, okuyinto linamathele amaseli lwegciwane. Isithako asebenzayo amuncwa umzimba ngesikhathi esifushane emisipheni yomzimba futhi iqala ukusebenza yayo elwa namagciwane.

Ezimweni eziningi, umuthi ibekezelelwe kahle, kodwa kungadala ukusabela nomzimba. Futhi, lo muthi ingasatshenziswa kusukela ekuzalweni. Ngenxa yale njongo kukhona uhlelo esikhethekile kubalwa umthamo. kabanzi kakhulu esetshenziswa-antibiotic emkhakheni wezilwane. Yena kusiza izilwane balahle namagciwane kulesetayelekile esiswini namathumbu.

Ngezinye izikhathi imithi "Gentamicin" kungaholela ukulahlekelwa kukuzwa, futhi lokhu ethile nendlela yawo ebanzi. Ngokutadisha zonke izibuyekezo, ikakhulukazi odokotela, ungabona indlela elinamandla ngayo izidakamizwa elwa namagciwane. It has a umsebenzi omkhulu ngokumelene anaerobic Gram-HIV futhi Gram-negative eziphilayo. I eziyinkimbinkimbi futhi engabelwe ekwelapheni ephathwa inyumoniya futhi meningitis. Kufanele banamathele ngokuqinile umthamo zomuthi ukuze ugweme engemihle. Ngokusho kochwepheshe abaningi, lesi sidakamizwa "Gentamicin sulfate" anobuthi. Ukusetshenziswa Its njalo angaphazamisa umsebenzi wazo zonke zomzimba. ejenti elwa namagciwane akufanele isetshenziswe ngaphandle kokubonisana onguchwepheshe.

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