ImpiloAmalungiselelo

Izidakamizwa "Mazeppa": yokusetshenziswa. Izibuyekezo sokulungiselela "Medazepam"

Kwezinye izimo, lesi sidakamizwa "Mazeppa" ingasetshenziswa? Inani, izinkomba kanye nemiyalelo zomuthi ethulwa ngezansi.

Ifomu, ukwakheka

"Mazeppa" - Tablets round, Valium. nempahla yabo eyisisekelo Medazepam. Ngokuphathelene izingxenye ezengeziwe, njengoba aphume ashone isitashi, monohydrate lactose ne-calcium stearate.

umphumela we izidakamizwa

Yiziphi amaphilisi, "Mazeppa"? Iziyalezo yokusetshenziswa Lithi kuyinto umenzeli anxiolytic, noma okuthiwa imijovo. Lesi sidakamizwa kuyinto esuselwe benzodiazepine. Liveza anxiolytic, antiepileptic futhi imisipha relaxant izici, futhi eliphuphile timolepticheskoe umphumela.

imiphumela Hypnotic futhi sine zomuthi siyenzeka ngezinga elincane kuka in ezivamile benzodiazepine anxiolytics. Kule ndaba, le nomuthi okukhulunywa siphathelene ehlukile iqembu "emini" zinhlungu.

Lokhu ejenti baxhumana receptor (benzodiazepine) limbic system, kanye kumiswa i brainstem Kuvuselela uplink (ubuchopho). Ngenxa yakhe iyona ukuvulwa iziteshi chloride okwagcina kuholela umphumela retarding ka Gaba ku CNS.

Phawula futhi ukuthi lesi sidakamizwa "MAZEPA", imiyalelo for ukusetshenziswa okuyinto kuchaziwe ngezansi, kusiza ukuqeda nokukhathazeka, ukucindezeleka psychoneurotic, ukukhathazeka, Uvalo nokukhathazeka eziphindaphindekayo jikelele motor ingqondo. Ngaphezu kwalokho, kuba kuzinze the NS autonomic, sivuselela similo sakhe ngekwemiva ukuhlolwa ezibucayi isifo sabo siqu.

kinetics

Yiziphi imingcele pharmacokinetic sici imijovo "Mazeppa"? Iziyalezo yokusetshenziswa ithi ngemva ukungenisa ithebhulethi ngokushesha ugxile inani 50-75%. ingqondo esiphezulu egazini safinyelela emahoreni amabili kamuva. Sesibopho ukuthobisa plasma-plasma amaprotheni 99,7%.

Metabolites zihlobene esebenzisa nezinso emathunjini amahora 20-175.

ubufakazi

Tablets "Mazeppa", ukubuyekezwa ozosithola ngezansi, esetshenziselwa ukucasuka, uvalo nevuso ukungezwani sezinzwa. It is ibuye Kunconywa ukusebenzisa izindlela at nokuqaleka kubantu abaphethwe ukuba umlutha wotshwala, ukuvimbela migraines kwabadala syndrome.

Ngo paediatrics lokhu izidakamizwa isetshenziselwa excitability anda wengane, lability engqondo futhi "isikole" nezifo zengqondo.

Izimo

Izindlela kuncike akufanele kuthathwe ngesikhathi sokukhulelwa, myasthenia gravis, "ebusuku" zokuphelelwa umoya medazepama ukungabekezelelani, pathologies ka kwezinso nesibindi, ukuncelisa nezinhlobo ezahlukene kuye (zezidakamizwa, utshwala). Ngaphezu kwalokho, izidakamizwa esebenzayo is contraindicated ku ataxia cerebellar, organic zokugula HC, umfutho ophakeme wegazi ocular, nokuvaleka kwemigudu yokuphefumula kanye ataxia umgogodla.

Imijovo "Mazeppa": yokusetshenziswa

"Medazepam" Tablets zithathwa kathathu ngosuku, eziqala umthamo ongaphakeme 5 mg. Kancane kancane inani inxusa kushintshwe 30 mg ngosuku. Ezimweni ezingavamile, zivunyelwe ukuba zithathe 40 mg zomuthi ngosuku.

Ngo-nesineke ukwelashwa Kunconywa ukuthi ukwelashwa uhlelo ezilandelayo: 5 mg izidakamizwa ekuseni 10 mg - kusihlwa. Kuleso sibhedlela kungase umthamo nsuku zonke esiphezulu sale ejenti senyukela 60-70 mg.

Isikhathi salesi ejenti kwelashwa izinyanga 2 (esiphezulu). Ngemva kwezinsuku ezingu-30, i-course kungaba liphindwe.

uhlangothi imihlola

Isihloko kungabangela imiphumela elandelayo:

  • dyspepsia, kukhuphuke bilirubin, AST, ALT, nomlomo owomile;
  • tachycardia, umfutho wegazi udedele;
  • stupor, disinhibition, ubuhlungu bekhanda, ukulahlekelwa amandla okukhumbula anterograde, yokuhlala paresis, ukucindezeleka, ukuba nesiyezi, dysarthria, ukukhathala, disorientation, ataxia, ubudlova, ukudideka;
  • kubantu abanegciwane COPD uma nithatha ebulilini zomuthi waphawula hypoventilation alveolar;
  • isimiso yaleli pheshana zokuphefumula kanye ukulimala kobuchopho waphawula okusithiyayo isikhungo zokuphefumula.

izincomo ezithile

Amaphilisi "Medazepam" kungase kube nomthelela kule ukuphazamiseka ukunakwa inkumbulo, kanye nokwehla ekufundeni.

Ndawonye nokusetshenziswa iziphuzo impermissible izindlela etanolsoderzhashih.

It income ukuhoxiswa kancane kancane izidakamizwa ekwelapheni nokuqaleka.

ukwelashwa okuqhubekayo kungasenza yakha imithi ukuncika medozepama.

Inani kanye nokubuyekeza

Izindleko ukucabangela imijovo kuba ruble ngu-150.

Nobufakazi ukukhombisa tolerability kuhle zomuthi kuhambisana yonke imiyalelo udokotela futhi senze njengoba siyaliwe nokushintsha kokudla nokufakwa. Nakuba ezimweni ezimbalwa lokhu kusho okwamanje ikhuthaza ukuluthwa izidakamizwa eziyingozi, ukuncishiswa potency, nokugcinwa urinary, ukusabela ayindida, komzimba nezinto, ubuhlungu besifuba kanye dysmenorrhea.

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