EzempiloAmalungiselelo

Yini esiza "Hypothiazid." "Hypothiazide": imiyalelo, ukubuyekezwa, ukufana

Namuhla sizokutshela ngalokho okusiza "Hypothiazid"? Futhi, ezintweni ezikulesi sihloko uzonikezwa imiyalelo ekusetshenzisweni kwalesi sidakamizwa, impendulo yabathengi, uhlobo lokukhululwa, izindawo nokunye okunye.

Incazelo yokulungiselela, ifomu, ukupakisha nokubunjwa

Yini esiza Hypothiazid? Ngaphambi kokuphendula lo mbuzo, kubalulekile ukutshela, ngaluphi uhlobo lo muthi oya kuma-pharmacy.

"I-Hypothiazide" iyatholakala ngendlela yamathebhulethi amhlophe (ingaba nomthunzi omnyama). Zinezakhiwo eziyindilinga, ezingozini kolunye uhlangothi nokuqoshwa "H" ngakolunye uhlangothi.

Isithako esisebenzayo salesi sidakamizwa i-hydrochlorothiazide. Ihlanganisa izinto ezisizayo ngesimo se-magnesium stearate, i-lactose monohydrate, i-talc, i-gelatin nesitashi sommbila.

Ekuthengiseni kwalo mkhiqizo kufika amabhulashini, ahlanganiswe emabhokisini amakhadibhodi.

Isenzo sempilo

Uyini umuthi "Hypothiazid"? Yini ewusiza lo muthi?

Ngokwemiyalelo, isidakamizwa esibuzwayo yisidakamizwa. Indlela eyinhloko yokwenza isenzo sokwanda kwe-diuresis ngokuvimbela ukubuyiselwa kabusha kwe-chloride kanye ne-sodium ions esifundeni sokuqala se-tubulus ye-renal. Lokhu kuholela ekunyuseni kwe-chlorine, i-sodium futhi, ngenxa yalokho, amanzi.

Kumele kuqashelwe ukuthi emva kokudliwa kwalesi sidakamizwa kwandisa ukukhipha kwamanye ama-electrolyte, noma kunalokho, i-potassium ne-magnesium.

Emithonjeni emikhulu yokwelapha, imiphumela ye-natriuretic neyesifo sezitho zomuthi zifana.

I-Diuresis ne-natriuresis zenzeka zingakapheli amaminithi angu-120 futhi zifinyelele inani eliphezulu emva kwamahora angu-4.

Kumele kuqashelwe ukuthi lesi sidakamizwa sinciphisa umsebenzi we-anhydrase carbonic ngokukhulisa ukuphuma kwama-bicarbonate ions. Kodwa-ke, lesi senzo sesidakamizwa sibuthakathaka futhi asithinti i- pH yomchamo.

Into esebenzayo "Hypothiazide" inezakhiwo ze-hypotensive. Kumele futhi kuthiwa ukuthi i-agent engumbuzo ayithinti ukucindezelwa kwegazi evamile.

AmaKinetics omuthi

Ingabe lesi sidakamizwa "Hypothiazid" sithatha? Imfundo, incazelo yombiko wezidakamizwa ukuthi i-hydrochlorothiazide ayitholakali ngokuphelele, kodwa ngokushesha inamathela ohlelweni lokugaya ukudla. Lesi senzo sihlala amahora angu-6-12.

Uma uthatha izidakamizwa ngaphakathi kumthamo we-100 mg, ukuphakama kwayo kwe-plasma kufinyelelwa emva kwamahora angu-2.5.

Ukuxhumeka kwamaprotheni e-plasma kungama-40%.

Ngokusho kochwepheshe, i-hydrochlorothiazide idonswa kanye nobisi lwebele futhi ingena emkhawulweni we-placental.

Leli remedy lidonswa izinso zingakapheli amahora ayisithupha.

Imithi: "Hypothiazid": yini ewusizo?

Leli thuluzi limiselwe:

  • Ukuvimbela ukwakheka ngamatshe emgqonyeni we-urinary kubantu abafakwe kule sifo (ngenhloso yokunciphisa i-hypercalciuria);
  • I-hypertension ye-arterial (ye-monotherapy futhi ihlanganiswe nezinye izidakamizwa eziphikisayo) ;
  • Ukulawulwa kwe-polyuria (ikakhulukazi isifo sikashukela se-nephrogenic esingekho ushukela);
  • I-Edematous syndrome yemvelaphi ehlukahlukene (i-premenstrual tension syndrome, i- nephrotic syndrome, ukwehluleka kwezintuthwane okungapheli, i-glomerulonephritis enamandla, ukwelashwa nge-corticosteroids, ukuhluleka kwenhliziyo okungapheli, ukucindezeleka kwe-portal).

Ukungafani

Cishe lokho, kusuka kulokho "Hypothiazid" kusiza, sitshele ngenhla. Kumele futhi wazi mayelana nokuphikisana kwalolu remedy. Zihlanganisa:

  • Izingane kuze kube yiminyaka emithathu;
  • Ukwehluleka okukhulu kwesinselo;
  • Anuria;
  • Ukuhluleka kwe-Hepatic ngezinga elibi;
  • Isifo sika-Addison;
  • Isifo sikashukela sinzima ukulawula;
  • Hypokalemia ephazamisayo, hyponatremia, hypercalcemia;
  • Ukuzwela okwedlulele ezingxenyeni zomuthi nezidakamizwa ze-sulfonamide.

Ngokunakekelwa okukhethekile, le nqubo kufanele isetshenziswe ku-IHD, hypokalemia, isibindi se-cirrhosis, i-hyponatremia, i-gout, i-hypercalcemia, i-glycosides yenhliziyo, ukubekezeleleka kwe-lactose kanye nabantu asebekhulile.

Isidakamizwa esithi "Hypothiazide": imiyalelo yokusetshenziswa

Ukubuyekezwa, ukufana kwezidakamizwa ezibuzwayo kuvezwe ekugcineni kwalesi sihloko.

Amathebulethi kufanele athathwe ngemuva kokudla. Umthamo wabo ukhethwe ngenkathi yokwelapha, ngabanye.

Ukuqalwa kokuqala kwesidakamizwa kubantu abadala:

  • I-syndrome yokuhlukunyezwa kwangaphambi komzimba: ukuthatha imithi iqala ngokubonakala kwezibonakaliso zokuqala ngaphambi kokuqala kokuya esikhathini (ngesamba sama 25 mg kanye ngosuku).
  • I-Edema syndrome yemvelaphi ehlukahlukene: 25-100 mg kanye ngosuku noma kanye ngezinsuku ezimbili. Ezimweni ezimbi, umuthi unqunywe ku-200 mg.
  • I-hypertension ye-arterial: 25-50 mg kanye ngosuku. Umphumela wokwelapha walesi sidakamizwa ubonakala ngaphakathi kwezinsuku ezingu-4.
  • Isifo sikashukela esingeyona isifo sikashukela nephrogenic: 50-150 mg ngosuku (ngezimpendulo eziningana).

Ngokuphathelene nezingane, kubo izidakamizwa ezibuzwayo zibekiwe ngokucabangela isisindo. Izinga lansuku zonke li-1-2 mg / kg.

Izenzakalo ezimbi

Manje uyazi ukuthi i-Hypothiazide iyasiza ngani. Ngokumelene nesimo sokuthatha le mithi, ukuphendula okuhlangene okulandelayo kungase kuthuthuke:

  • I-Anorexia, umlomo owomile, ama-cramp muscle, isifo sohudo;
  • Ubuhlungu emisipha, ukuqotshwa, ukukhathala, i-cholecystitis, ubuthakathaka, i-jaundice ye-cholestatic;
  • I-Lethargy, i-pancreatitis, ukoma, i-sialadenitis;
  • I-arrhythmia, i-anemia ye-aplastic, i- vasculitis, i-thrombocytopenia, ikhanda, i-leukopenia;
  • Isizungu, i-hemolytic anemia, ukuphazamiseka kwezinso zokusebenza, i-agranulocytosis nabanye.

Ama-analogues nezibuyekezo mayelana nomuthi "Hypothiazid"

Ukubuyekezwa kwe-"Hypothiazide" kubika ukuthi lokhu kuyisimo se-diuretic esisebenzayo futhi esheshayo. Ukudla kwamathebulethi anjalo kuvimbela ukwakheka kwamatshe emgqeni we-urinary, kuncishisa ukucindezeleka kwegazi futhi kuqede ukuvuvukala kwemvelaphi ehlukahlukene.

Ububi besidakamizwa esibuzwayo bubandakanya inani elikhulu lokuphendula okubi.

Izidakamizwa ezifanayo zalesi sidakamizwa ziyi: "Hydrochlorothiazide", "Hydrochlorothiazide-SAR", "Dichlorothiazide", "Hydrochlorothiazide-Verte" nabanye.

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