ImpiloAmalungiselelo

"Brilint": incazelo izidakamizwa, imfundo. Analog "Brilinta"

"Brilint" - umuthi okuyinto kabanzi ezisetshenziswayo ekuhlinzeni nezenhliziyo, njengoba has ankoagulyantnym nemiphumela antiplatelet. Ezimweni eziningi, usetshenziselwe injongo cupping angina (engazinzile ifomu) nobuhlungu ischemic, kanye ejenti prophylactic ngokumelene ukopha ngokushesha ngaphambi nje kokuba ahlinzwe.

Sakhiwo Ukwakheka

Iyatholakala "Brilinta" 90 mg (futhi analog) amaphilisi. Basuke embozwe ikhava ifilimu ka abe luhlaza aphuzi. Umumo round biconvex.

The main isithako zomuthi kuyinto ticagrelor. Phakathi adjuvants ihlaba umkhosi:

  • mannitol;
  • magnesium stearate;
  • calcium hydrogenphosphate;
  • sodium carboxymethyl isitashi;
  • giproloza.

Le filimu, esikhundleni salokho, kantsi sicuketse loku hypromellose, talc, ama-titanium dioxide, macrogol, udayi (ophuzi oxide).

Umthelela eyinhloko izidakamizwa

"Brilint" has antiplatelet isinyathelo, isb kuvimbela wokuhlanganisa amahlule. Ngenxa yalokho main asebenzayo izidakamizwa ingxenye - ticagrelor - platelet balahlekelwe ikhono banamathelane, futhi ngaleyo ndlela yakha amahlule.

Ukuhlola okuhlukahlukene uqinisekise yokuthi indlela "Brilinta" ngempumelelo ngaphezulu lihambisana salicylic acid. Analogichinye ukwamukelwa futhi mayelana Analogue "Brilinta" - "Plavix". Kulezi nokulingwa abathintekayo iziguli isifo senhliziyo ngo eyehlukene, futhi kubonelelwe isisindo sabo, ubulili.

Umgomo oyinhloko wabo yokwelapha usebenzisa umkhiqizo wathi - ukunciphisa ingozi yokufa, okungase kubangelwe ukungasebenzi esimiso senhliziyo nemithambo yegazi, ikakhulukazi pectoris angina futhi isilethikusebenza.

izinkomba

Reception "Brilinta" kuboniswa esimweni isidingo ukunciphisa igazi ekunqandeni, kuhlanganise nokuvinjelwa yezinkinga yokuthola izifo eziphathelene nenhliziyo ngesimo thrombosis futhi thromboembolism. Yingakho lolu izidakamizwa kuboniswa ngenxa:

  • angina engazinzile (Lokhu zokugula libhekene Ukuwohloka kwegazi igazi ukuze imisipha yenhliziyo, okuyinto okusongelayo esivimba amanzi);
  • isilethikusebenza (kokufa ingxenye inhliziyo);
  • enza imisebenzi kuhlinzwa ezitsheni yenhliziyo of imisipha yenhliziyo (ngesikhathi ukungenelela yenhliziyo percutaneous, noma yenhliziyo Umthambo ukuhlinzwa dlula).

Ngaphezu ubufakazi ngqo, ukuze "Brilint" ngokubona udokotela angaqokwa ukuze kuncishiswe thrombosis kwezinye izimo zokucabanga okubangelwa isifo, njengalapho dissemirovannom coagulation intravascular.

Izimo

Kunezindlela eziningana ukulinganiselwa, lapho ukusetshenziswa "Brilinta" akuvunyelwe. Lezi zihlanganisa:

  • isici esiyingqayizivele, kuhlanganise hypersensitivity kuya izidakamizwa esebenzayo noma okungenani eyodwa koponentu ezengeziwe;
  • ukopha asebenzayo, sithwele sokugembula;
  • haemorrhagic unhlangothi ukuma ukuthi washukumiseleka ngaphambili;
  • wehlise umsebenzi hepatocyte, ngokumelene okwenzeka yokwehluleka kwesibindi ukusebenza;
  • ukuphatha izidakamizwa, isenzo eyinhloko esakhiwa ngo okusithiyayo of enzyme CYP3A4 ( «clotrimazole," "Ritonavir", "nefazodone");
  • Izingane ezineminyaka engu-18;
  • phakathi nokukhulelwa kanye lactation.

In the ukungabikho Izimo kudingeka wenze ngaphambi kokuqala ukwelashwa nale izidakamizwa.

Yokusetshenziswa

Thatha "Brilint" kufanele kube ngaphakathi lonke, umuthi akumele ezokuhlafunwa. Ukusebenzisa izidakamizwa kuzimele isikhathi ukudla. Tablets ziphuze esincane ketshezi.

Isikali ezinconyiwe: 1 tablet ngosuku. Kubalulekile ukuthatha imithi nsuku zonke ngesikhathi esifanayo.

Inkambo yokwelapha nokusetshenziswa "Brilinta" (esikhundleni zingenziwa eside) kufanele uqale nge umthamo double (amaphilisi amabili ngosuku lokuqala), bese ukuthuthela umthamo owodwa we-90 mg. Endabeni yokwamukelwa zomuthi akufanele zisebenzisa umthamo double. Ngakusasa ngemva qhuba aphuthelwe reception evamile "Brilinta." Nokho, kufanele izimo ezinjalo kugwenywe.

Isikhathi isilinganiso ukwelashwa - ezingu-12.

Ngaphezu kwalokho, watusa kanyekanye acetylsalicylic acid.

side effects

Phakathi ukubonakaliswa atypical ethola avelele:

  • ukunciphisa engahlula ka igazi ekunqandeni ukuthuthukiswa ukopha okungavamile;
  • komzimba;
  • isicanucanu;
  • ukuhlanza.

Lapho imiphumela emibi izidakamizwa kufanele simiswe ngokushesha.

ukweqisa izidakamizwa

Endabeni zimpawu ezilandelayo kungenzeka kokuthola ngemithamo okwandisiwe izidakamizwa:

  • isicanucanu;
  • ukuvuvukala;
  • ukopha;
  • ukuphazamiseka inhliziyo.

Lapho kwenzeka kumelwe ayeke ukuthatha izidakamizwa, ukuba lavage esiswini, amathumbu, futhi ukwelashwa lingaze.

analogs

Ngezinye nakwenzeka ngokuthatha izidakamizwa kudingeka azi ukuthi esikhundleni "Brilintu". Phakathi nozakwabo eziba sobala:

  1. "Zilt". Lokhu Analogue "Brilinta" intengo lihlukile, kodwa imiphumela kokubili izidakamizwa zifana futhi ezihlose nokuvimbela thrombosis. isithako esebenzayo clopidogrel. I izinkomba ngoba ukusetshenziswa kwezimali kukhona isilethikusebenza, yenhliziyo syndrome, isifo sohlangothi, fibrillation atrial, yenhliziyo isifo Umthambo okklyuizonnaya. "Zilt" elinesimo ezingavamile side effect.
  2. "Plavix". "Brilinta" noma "Plavix" - okuyinto engcono? Ithi neze. Le mithi zihlukile izidakamizwa esebenzayo, kodwa umphumela banayo efanayo. Lokhu kuvumela kokuma Yiqiniso yokwelapha is enye indlela uqhubeke nokwelashwa nomunye. Analogue "Brilinta" "Plavix" inikezwe iziguli imihlola atherosclerotic ezikhonjwe, iziguli ngemva kokushaywa yinhliziyo kanye nesifo sohlangothi. Lokhu umuthi analog futhi ashibhile. Yini ukukhetha: "Brilinta" noma "Plavix". Yikuphi okungcono? Tshela udokotela.
  3. "Lopirel". Lokhu Analogue "Brilinta" wenza ngesisekelo clopidogrel, yingakho isenzo siqondiswe zegazi, ukuvimbela nabo banamathelane. Ngokungafani nezinye izindlela, "Lopirel" kungathinta ukusebenza kwemizwa, zokuphefumula, uhlelo zemisipha, kanye hematopoiesis. Ngaphezu kwalokho, Kuhle ukukhumbula ukuthi lokhu Analogue izidakamizwa "Brilinta" akuyona yokuqala, futhi ejwayelekile, okungukuthi ikhophi "Plavix".

Ngaphezu kwalezi analogue avunyelwe ukusetshenziswa nezinye izidakamizwa ukuthi ube nomphumela ofanayo, kodwa kuhluke indlela yesenzo ( "Cardiomagnyl", "Aspekard", "aspirin-Cardio").

Imigomo nemibandela isitoreji

Impilo "Brilinta" (amazwana ngawo ngaso sonke positive) uneminyaka engu-2. Ngakho kubalulekile ukuba bagcine umbuso lokushisa (egumbini lapho ejenti egcinwe kufanele kube degrees ngaphansi kuka 30, kufanele kube khona ukukhanya nomswakama). Ngaphezu kwalokho, ithuluzi kufanele bavikeleke izingane.

Khumbula ukuthi wonke ama-aphoyintimenti kufanele ukuqhuba udokotela.

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