ImpiloAmalungiselelo

"Amantadine": yokusetshenziswa, analogs, ukubuyekezwa

Umuthi 'Amantadine "libhekisela namagciwane futhi antiparkinsonian. Ngenxa imiphumela evelele ku isimiso sezinzwa esiyinhloko phambi ethatha kumele ayejwayele Izimo, kanye uthole ukuthi yini imithi yakhe akufanele kuhlangene. Ngokuvamile, izidakamizwa ezinqunyiwe ekwelapheni isifo i-Parkinson e ukwelashwa. I kuyaqabukela asetshenziswa njengenhlangano agent elwa namagciwane. Ngokuvamile ukhetha nezinye izidakamizwa ukuthi ifa okumbalwa imiphumela engemihle.

Kanjani imisebenzi izidakamizwa?

Isenzo "Amantadine" okuhloswe ngaso glutamate receptor. Ngenxa enciphile yabo Ukuvinjwa nomthelela ukuntula striatum Dopamine ngemuva - umphumela antiparkinsonian ngakho abayifunayo. Umthelela namagciwane ukuthi izidakamizwa kuvimbela Ukungena igciwane (Umkhuhlane A) kumaseli izicubu zomzimba.

Umzila yokuphathwa - ngomlomo. Okulandelayo "Amantadine" ugxile ipheshana wokugaya ukudla bese ufaka ekusakazeni igazi, lapho emakamu esiphezulu waphawula ngemva 4 amahora. Kufanele kuqashelwe ikhono zomuthi ukungena ngokusebenzisa isithiyo esinomhlapho, okuyinto ine umphumela emibi embungwini. "Amantadine" (yokusetshenziswa - ngezansi) is contraindicated hhayi kuphela kwabesifazane abakhulelwe, kodwa futhi ngesikhathi ibele.

isakhiwo

Isithako esebenzayo amantadine sulfate, kodwa kunezinye izingxenye asizayo ngo kwengoma. Bona ikakhulukazi kufanele sinake uma kukhona ukusabela nomzimba. Ukulungiswa iqukethe lactose monohydrate, gelatin, talc, isitashi kanye cellulose. Futhi kule - magnesium stearate, Silicon dioxide futhi titanium, polyethylene glycol.

Uma sisetshenziswa "Amantadine"?

Lesi sidakamizwa engabizi namagciwane asetshenziselwa ukwelapha Umkhuhlane A, kanye nokuvinjelwa. Ngaphezu kwalokho, ukusebenza ezimise okwama-tile (ibangelwa igciwane ke Herpes zoster) ukwehlisa neuralgia. Okunye okubonisa - parkinsonism.

"Amantadine": yokusetshenziswa

Indlela ukuthatha izidakamizwa? Tablets "Amantadine" (intengo kuncike endaweni sokuthenga -. Ruble 130-150) Kunconywa ekuseni, njengoba kungase kube kusebenze ngokweqile isimiso sezinzwa esiyinhloko, futhi ngenxa yalokho, okuvela kuyo ukuqwasha nezinye imiphumela emibi (nesiyezi, ikhanda). A umthamo owodwa kuxhomeke isifo futhi umphumela oyifunayo. Okunqumayo kuphela udokotela ukuba khona ikhumbula izici ngamunye isiguli kanye kunjalo emtholampilo. Ngo parkinsonism ngesonto lokuqala, ngokuvamile iqondiswa mg 100 zomuthi ngosuku, futhi ngemva okwandisa umthamo (esiphezulu - 400 mg).

Loluhlelo ukwelashwa kushintshwe kuncike ekutheni izifo lesiguli ahlobene, ezifana nokwehluleka ukusebenza kwezinso lapho usukhulile futhi umthamo kumele kungancipha. Ukuze ngizwakalise anti-Parkinson umphumela umuthi kuhlangene nezinye izidakamizwa. Monotherapy kuyinto ayizwakali. Akufanele yini evele ukuziyeka izidakamizwa, njengoba kukhona ingozi Kucinisa izimpawu Parkinson kuze kube zinhlekelele akinetic. Lokhu kunjalo, ikakhulu bokucatshangelwa lapho uzingela abalulekile side effects - ukwenqaba imithi kumele ibe bushelelezi, kancane kancane kuyancipha umthamo.

ukwelashwa elwa namagciwane kuhilela ukuthatha imithi njalo ngemva kwamahora angu-12. Ngokuvamile, udokotela ekunika yokwamukela 1 tablet (100 mg), kodwa umthamo ephansi (nsuku zonke esiphezulu - 100 mg) ngoba iziguli esezikhulile. Ukwelashwa kufanele waqala ngokushesha lapho kuqala izimpawu, Inkambo yokwelashwa ngokuvamile izinsuku 5. Ukuze zokuvimbela kufanele uthathe 100 mg / ngosuku, ubude ekuphathweni ivela 2 kuya ku 4 amaviki.

Ukwelashwa nokuvikelwa neuralgia, kubangelwa H. zoster, sihlala 14 izinsuku bese uqalisa ukwelashwa kufanele kube ngokushesha ngemva uphethwe.

side effects

"Amantadine" (yokusetshenziswa - kwikhithi) has a uhlu enkulu yemiphumela emibi ngenxa ngokuyinhloko ikhono layo ukuze zingene kusivimbeli gazi ebuchosheni futhi kuthinte isimiso sezinzwa esiyinhloko. Phakathi kwabo - izinkathazo, ikhanda kanye isiyezi, ukuyaluza sezinzwa, amaphupho amabi, ukusangana (ezingavamile). Ngokuvamile kukhona inattention futhi ukudideka, ngakho kwesikhathi yokwelashwa, "amantadine" akufanele ukushayela izimoto futhi enze umsebenzi oyingozi okudinga ukuba agxilise ingqondo okusezingeni eliphezulu. Eminye imiphumela emibi - leukopenia, isicanucanu, uhudo, micturition kahle, ukuqubuka kwesikhumba, edema (ikakhulukazi in iziguli congestive senhliziyo).

Izimo

Ngaphambi kokuthatha lesi imithi, kufanele ubuyekeze ngokucophelela uhlu Izimo. Phakathi kwabo:

  • yokungezwani komzimba ukuze yezingxenye;
  • ukwehluleka kwezinso;
  • peptic isilonda isifo;
  • isithuthwane;
  • Ukukhulelwa ibele.

Yimiphi imithi angeke kuhlanganiswe "Amantadine"?

Umuthi ngokuvamile kuhlangene izidakamizwa anticholinergic namanye amanxusa ukwelapha isifo i-Parkinson, kuyilapho kukhona mutual ukuqinisa ukusebenza. Nokho, it is hhayi Kunconywa ukuba sihlanganise le ukulungiselela kanye "L-dopa", njengoba kukhona ingozi Kucinisa isinyathelo isimiso sezinzwa esiyinhloko (sengqondo, ukuhhema, amaphupho amabi). Ngesizathu esifanayo, "Amantadine" ungathathi esifanayo ukuze "Memantine".

Kuyadingeka ukuba senqabe utshwala, njengoba lokhu kuhilelani beqinisa imiphumela anobuthi phezu CNS. Futhi-ke ayifakiwe kanyekanye reception "amantadine" isisu, ngoba kulesi simo ephukile excretion namagciwane ejenti, futhi ngenxa yalokho, emakamu yayo egazini ongafinyelela amazinga ayingozi.

"Amantadine": nozakwabo. Yini ebaluleke ukuthenga?

Phakathi kwezidakamizwa kabani Ukwakheka nomongo asebenzayo kuhlanganisiwe amantadine (yokusetshenziswa analogs ezahlukene) kungenziwa isehlane, "PC-Merz" futhi "Neomidantan". Kugcine ekhishwe ngesimo gelatin amaphilisi egcwele powder emhlophe. "PK-Merz" - amaphilisi i igobolondo orange. Uhlu izinkomba kule nokulungiselela ebanzi. "PK-Merz" lisetshenzisiwe nangokuqondene kuhlasimulise okulimala ebuchosheni, ukudakwa endogenous, unhlangothi, ukuwohloka, chorea Huntington sika.

Izibuyekezo

Ngokwe kodokotela kanye neziguli, umuthi ihlinzeka umphumela evelele zokwelapha ngesikhathi esifushane. Ngokwe ukuya ikhambi amagciwane uphawu ngcono ngokushesha kahle. Phakathi imiphumela emibi ngokuvamile baphawula injabulo kwemizwa nokunakwa neziyaluyalu, kanye nezinye ezingavamile. Odokotela abaningi e parkinsonism ibhekwa kuya ukwelashwa njengoba Kunconywa "Amantadine", ukubuyekezwa ngokuvamile ikakhulukazi omuhle ngakho. Nakuba yimuphi izidakamizwa kukhona abaphikisi.

"Amantadine" - engabizi ejenti elwa namagciwane, okuyinto lungasetshenziswa e parkinsonism. Ngaphambi isicelo, qiniseka ukuthi uxhumane uchwepheshe, ngubani, banikezwe izici umzimba, futhi comorbidities, khetha umthamo edingekayo noma ukunikela noma yimuphi nezinye izidakamizwa ne nomphumela ofanayo.

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