ImpiloAmalungiselelo

"Flyuanksol": yokusetshenziswa, odokotela yangempela. Imiphumela emibi "Flyuanksola" analogue zomuthi

Uyini izidakamizwa "Flyuanksol"? Yokusetshenziswa zomuthi, izithako zako, imiphumela emibi, ifomu ukukhululwa kanye izakhiwo kwemithi zichazwe ngokuningiliziwe kulesi sihloko. Kusukela ke uzofunda ukuthi contraindications izinkomba akushilo izidakamizwa, ukuthi kubiza malini, kuzokwenzekani uma ukweqisa izidakamizwa, nokunye. D.

Ukwakheka izidakamizwa futhi ukukhululwa buyisiphi

Uyini umnyombo asebenzayo iqukethe imithi "Flyuanksol"? yokusetshenziswa imfundo nomuthi uthi njengoba ingxenye esebenzayo ke kuphuma hydrochloride flupenthixol.

Njengoba uhlobo ukukhululwa, kodwa namuhla kuyindlela kungatholakala kuphela amathonsi, amaphilisi kanye isixazululo, amafutha-based, senzelwe abaphathi esicutshini. Umuthi wokuqala ithunyelwa ingilazi zatemennom 10 ml, owesibili - e ibhokisi 100 noma 50 nowesithathu - ku ampoules yizicucu 10.

izakhiwo Jikelele zomuthi

Kungani imithi "Flyuanksol"? Nobufakazi ngalokhu izidakamizwa ethulwa ngezansi. Amaphilisi kanye umjovo iqembu antipsychotics. They possess anxiolytic, antidepressant nomphumela okulalisayo. okubuyayo ngalokhu izidakamizwa aqukethe ulwazi ukuthi kahle isebenze isimo esingokomzwelo isiguli futhi ubangela lithathelwe nomphakathi.

Izimfanelo kwemithi zomuthi

Yiziphi izici izidakamizwa kwemithi "Flyuanksol"? Yokusetshenziswa busikisela ukuthi leli izidakamizwa kuyinto neuroleptic, ivimbela receptor adrenergic futhi Dopamine zemizwa ingqondo. Ngenxa yalokho we ketshezi esebenzayo kufinyelelwa ukupholisa. Ngokuvamile, lokhu kwenzeka phezu sokuphuza isilinganiso esengeziwe somuthi njalo ngosuku-8.

Yini iziguli ngemithi "Flyuanksol"? Izibuyekezo iziguli aqukethe ulwazi oluningi ezithakazelisayo. Ezimweni eziningi, bona wazi ukuthi izidakamizwa esikhundleni ngokushesha aqede izimpawu sengqondo nokucindezeleka, kanye kunomthelela ukubuyiselwa ukucabanga. Iziguli ababe iziyaluyalu 'idla yodwa, kukhona nobudlelwano bese ukuzivumelanisa umphakathi.

Izici imithi

Kanjani lesi sidakamizwa "Flyuanksol"? Uphenyo kodokotela nabanye ochwepheshe bathi isici sale izidakamizwa wukuthi, kuncike umthamo kungaba isinyathelo isiguli ngezindlela ezahlukene.

umphumela Antipsychotic ububonisa emva isicelo nomuthi kusho i inani 3 mg ngosuku. By the way, ukushuba umthelela kwandisa ne umthamo.

Inani 25 mg ngelanga izidakamizwa akunamthelela sine. Nokho, kufanele kuphawulwe ukuthi ngesikhathi ngemithamo ephakeme, umuntu angaba sine imiphumela non-ethize.

Esikhathini umthamo ububanzi ogunyazwe neuroleptic kunomphumela evelele anxiolytic. Lapho usebenzisa i-ngemithamo emincane (kufika ku-3 mg ngelanga), umuthi angase bayisibonelo imithi ezivamile antidepressant.

Ngakho, lesi sidakamizwa "Flyuanksol" uyakwazi ukunciphisa izimpawu eyinhloko sengqondo, kuhlanganise okuyize paranoid, ukubona imibono engekho wacabanga sifo. It has izakhiwo disinhibitory (isb Kuvuselela futhi antiautisticheskim) futhi kunciphisa kwemizwelo, okwagcina ikhuthaza ukusebenza iziguli izimpawu futhi bacindezeleke, lithathelwe yabo yezenhlalo kusiza futhi sithuthukisa sociability.

Okuningi mayelana ifomu nemijovo

Ukulungiselela "Flyuanksol Depot" kuyinto isixazululo uwoyela senzelwe esicutshini edepho imijovo. Ngamanye amazwi, lokhu izidakamizwa imali ifomu flupenthixol.

Uma usebenzisa lokhu isixazululo ngemithamo amancane naphakathi (kufika ku 100 mg zonke izinsuku ezingu-14) esigulini akuyona ukupholisa unspecific. Nakuba-ke usakhula at ebulilini.

Yini ochwepheshe abathi mayelana leli fomu zomuthi ( "Flyuanksol Depot")? Izibuyekezo ukunikeza ukuthi ikhambi elinjalo has a ubude eside ukuchayeka isiguli, kunokuba amaphilisi imithi. Ngaphezu kwalokho, sibonga kuye, kulula lokufeza ukwelashwa okuqhubekayo antipsychotic, okuyinto ebaluleke kakhulu ezigulini musa afeze kadokotela.

Ngokwalokhu okungenhla kungenziwa baphetha ngokuthi izidakamizwa "Flyuanksol Depot" uyakwazi ukuvimbela umuntu uyahluleka uma elwa njalo elihlobene ne kokuphazamiseka nokuguqulwa yokwelapha. uyijova esicutshini kungaba kwenziwe ngezikhawu amasonto amabili noma amane.

Pharmacokinetics

amaphilisi baye ugxile isikhathi esingakanani "Flyuanksol"? Ngemva kokuphathwa temlomo emakamu esiphezulu element asebenzayo kufinyelelwa ku amahora mayelana 3-7 e-plasma. I bioavailability zomuthi 40%.

Active izidakamizwa isici kancane ingena isithiyo esinomhlapho. Kufanele kuphawulwe ukuthi, ngesilinganiso esincane, kuqokonyiswe nge ubisi lukamama. Phela, lo metabolites unomsebenzi neuroleptic.

kanjani umjovo "Flyuanksol Depot"? Umhlahlandlela ithi ngemva ujove esicutshini lomcebo cis (Z) decanoate -flupentixol asitholayo cleavage (enzymatic). Loku element asebenzayo we cis (Z) -flupentixol futhi decanoic acid. Ubuningi esiphezulu e serum kufinyelelwa lokuqala ekupheleni ngesonto lokuqala emva umjovo.

Lapho ethola izibhebhe ku zizalela inkathi yabo amahora angaba ngu-35. Uma yasetshenziselwa khona isixazululo umjovo, emakamu incipha exponentially kule serum (emva amasonto 3).

Kuboniswa nomuthi asebenzayo ngesimo metabolites ngokusebenzisa emathunjini, nezinso.

Izinkomba ukusetshenziswa ejenti neuroleptic

Kwezinye izimo, umuthi kubonisa "Flyuanksol"? isenzo sayo zingase zihluke, kuncike umthamo.

Umuthi kubonakala ngemithamo kuze 3 mg ngosuku izimo zokucabanga okubangelwa isifo ezilandelayo:

  • ukucindezeleka oluncane kanye degree ngokulinganisela, ephelezelwa ukukhathala, ukukhathazeka kanye nokuntuleka isinyathelo;
  • iziyaluyalu zengqondo abonisa ukusabela asthenic;
  • iziyaluyalu Neurotic (ezingamahlalakhona), ephelezelwa nokunganaki, ukucindezeleka nokukhathazeka;
  • ne-acute nesimo yokukhathazeka, kanye isimo ukucindezeleka ngokweqile ngokomzwelo, angadingi sine noma umphumela okuyiluthayo (isibonelo, uma isiguli zingahlukumezi zinhlungu).

Nomuthi "Flyuanksol", analogue zazo izokwethulwa ekupheleni isihloko, umiswa at imithamo 3 mg ngelanga nokuningi uma kukhona ukuphambuka kulokhu okulandelayo: Izimo ingqondo ukuthi ahambisana okuyize Paranoid, ukuhhema, ukuphazamiseka ukucabanga, anergy, abantu abaningi abasinaki futhi akakhulumi.

Izimo ukusetshenziswa ejenti neuroleptic

Kwezinye izimo, it is hhayi Kunconywa ukusebenzisa izidakamizwa "Flyuanksol"? Yokusetshenziswa zihlanganisa uhlu olandelayo Izimo:

  • ubudala zezingane (iminyaka engu-18);
  • CNS nokucindezeleka;
  • lactation;
  • ngesikhathi sokukhulelwa;
  • ukudakwa (acute) barbiturates;
  • igoqe;
  • ukudakwa acute opioid analgesics;
  • pheochromocytoma;
  • oludakayo ubuthi acute;
  • uthi comatose;
  • umnkantsha ukucindezelwa;
  • izinguquko sokugembula egazini;
  • hypersensitivity kuya neuroleptics kokuba isakhiwo tioksantenoviy.

Kufanele kuqashelwe ukuthi akutuseki linqume izidakamizwa ngemithamo emincane (kuya ku-3 mg) esimweni hyperactivity noma excitations.

Izidakamizwa "Flyuanksol": imfundo (amaphilisi, lehla)

Ukuze ekwelapheni nokukhathazeka futhi bacindezeleke iziyaluyalu umthamo kokuqala nomuthi e izibhebhe kufanele kube 1 mg kanye ngosuku (mhlawumbe ekuseni), noma 500 mcg kabili ngelanga. Uma umphumela zokwelapha engekho, inani izidakamizwa ngeviki zingandiswa 2 mg. Ngakho umthamo wansuku zonke (2-3 mg) ihlukaniswe izigaba eziningana. Uma umphumela engekho uma usebenzisa izidakamizwa ku umthamo maximal (ngamanye amazwi, 3 mg), khona-ke kufanele uyekwa.

Ekwelapheni izimo ingqondo setha inani imithi ngamunye kuphela. I kokuqala umthamo nsuku zonke kufanele kube 3-15 mg 3 ngemithamo ahlukaniswe. Uma wayefisa, ivolumu wathi zingandiswa kuya ku-20 noma-30 mg ngosuku. Umthamo esiphezulu akufanele bube ngaphezu kuka-40 mg.

Njengoba emelelwa ukwelashwa yesondlo ejenti iqondiswa i inani 5-20 mg kanye ngelanga (ekuseni).

Ngokuqondene iconsi "Flyuanksol", kufanele kuphela ayiswe. Odokotela bavame linqume izidakamizwa kuleli fomu kuphela icala uma, nganoma isiphi isizathu, awukwazi ukuthatha imithi ngomlomo (tablet). Isikali eyeseka iziguli kuyinto 4-40 mg ngosuku.

Ukufakwa "Flyuanksol": imfundo, ukubuyekezwa nesineke

Isixazululo oily ngoba esicutshini edepho imijovo kumele iqondiswa ezijulile waya engxenyeni engenhla elingaphandle ezinqeni. Isikali nezikhawu phakathi ukwelashwa kufanele zifakelwe kuphela ngamunye (ezimele nomphumela oqabulayo).

Lokhu ekwakhiweni ngokuvamile lisetshenziswa isamba 20-40 mg (noma 1-2 ml) njalo emavikini 2 noma 4. Kufanele kuqashelwe ukuthi ezinye iziguli kungadinga imithamo emikhulu nezikhawu esifushane phakathi imijovo.

Uma umthamo eziqokiwe yokwelapha umjovo (20 mg / ml) ingaphezu 2 noma 3 ml 1 inqubo, kubalulekile ukuba siqhubeke ne isixazululo emakamu eliphezulu.

Ukulungiselela 100 mg / ml kufanele injected volume of 50-200 mg (noma 0.5-2 ml) njalo emavikini 2-4. Ngo lokubuya kwesifo oyingozi noma exacerbation lesi sifo ngezinye izikhathi sidinga wesikhathi esisodwa isingeniso kusho e isamba kuze kufinyelele 400 mg ngezikhawu ngesonto 2 noma 1. Ngemva izimpawu acute ukudlula, kumele ukukhiqiza ukuncipha kancane kancane umthamo kumuntu yesondlo (20-200 mg njalo emavikini 2-4).

Uma kudingeka ukuba kudlule ifomu ngomlomo kwezidakamizwa parenteral ukulungiselela yokwelapha osekelayo, kutuswa ukuba kusekelwe uhlelo ezilandelayo:

  • Inani nsuku zonke (e mg) kwezidakamizwa e izibhebhe x 4 = umthamo owodwa (e mg) umjovo zonke izinsuku ezingu-14.

Kufanele kuphawulwe ukuthi kungakapheli isonto elilodwa emva nokuphathwa izidakamizwa belulekwa ukuba baqhubeke nokuphuza lo muthi amaphilisi, kodwa umthamo ephansi. Landela-up ivolumu kanye igebe phakathi emileyo ngokuhambisana nomphumela oqabulayo.

Isikali Maximum isixazululo komjovo (owodwa esigabeni) imayelana 400 mg. Ngakho igebe phakathi imijovo kumele okungenani ngesonto.

Ngokusho izimpendulo iziguli, uma isetshenziswa kahle, ukulungiswa kanye nokubhekela izincomo yezokwelapha, it has a nethonya elihle esimweni sazo jikelele ngokomzwelo.

side effects

Can ibe nomphumela ongemuhle umuthi emzimbeni "Flyuanksol"? ukungaphathwa kahle imithi kuba khona izidakamizwa, kungakhathaliseki injalo. Lapha abayikho manje.

  1. isimiso sezinzwa: giperkinetiko-abanomfutho wegazi ophakeme syndrome (ukukhanya extrapyramidal), ubuthakathaka, akathisia, ukutubeka komzimba, isiyezi, lengqondo retardation, dyskinesia tardive, ukusabela dystonic futhi neuroleptic syndrome ebulalayo.
  2. Inhliziyo negazi izitsha: tachycardia, hypotension, orthostatic.
  3. uhlelo hematopoietic: granulocytopenia.
  4. Izinzwa: ukuphazamiseka yokuhlala.
  5. GI: ukuqunjelwa, jaundice cholestatic, nomlomo owomile, izinguquko lezivakashi e umsebenzi ukuhlolwa isibindi.
  6. Endocrine uhlelo: kwesisindo galactorrhea, ukujuluka, gynaecomastia, ubuthakathaka, dysmenorrhea, isifiso sokudla kakhulu, kwehle libido, ukushisa komzimba.
  7. uhlelo urinary: nokugcinwa urinary.
  8. Komzimba: dermatitis, photosensitivity, futhi ukuqubuka kwesikhumba.

imiyalelo Special ukusetshenziswa

Nge imithi ngokucophelela okukhulu elibekelwe iziguli ezinokuphazamiseka zenhliziyo, iziyaluyalu convulsive, nokuvaleka kwemigudu yokuphefumula, ukufiphala kwamehlo Parkinson, izilonda esiswini namathumbu 12-tiperstnoj, isifuba somoya, ukuba umlutha wotshwala, emphysema, nokugcinwa urinary, yokwehluleka kwesibindi, futhi ingozi Hyperplasia Prostatic.

Uma isiguli kwake wathola neuroleptics noma tranquillizers nge nomphumela okulalisayo, kubalulekile ukuziyeka ngokushelela.

Lapho ukwelashwa eside, ikakhulukazi imithamo ephezulu Kunconywa ukulawula kanye nokulinganisa isimo lesiguli ukuze ulungise yesondlo umthamo.

Ekwelapheni kanyekanye lwesabelo sikashukela ka wathi ekwakhiweni kungadinga ukulungisa lemali we-insulin.

Ngo ukusetshenziswa neuroleptics angagcina neuroleptic syndrome ebulalayo. Izimpawu zayo eziyinhloko imisipha rigidity, komzimba, isimo ezishintshwe engokwengqondo ukungasebenzi kwekhono autonomic nesimiso sezinzwa. Lapho izimpawu ezinjalo zidinga yokukhansela ophuthumayo ukuqokwa izidakamizwa kanye nokwelashwa bangisekela lingaze.

Ezimweni eziningi, imithi "Flyuanksol" akakubangeli ukupholisa. Kodwa, naphezu kwalokhu, kubalulekile ukuba acabangele ukukhinyabezeka kwayo nebangomuso ikhono usebenze umshini ngokuphepha, noma ezinye izindlela. Ngizothanda futhi ukuba uqaphele ukuthi ngesikhathi therapy (ikakhulukazi ekuqaleni), iziguli kufanele ugweme umsebenzi ezinobungozi (ukunquma indlela abantu abasabela ngayo izidakamizwa).

amacala ukweqisa izidakamizwa

Uma imithi esithathwayo kahle (izwi elithé ukuphakama), kungase kwenzeke yokweqisa. Kulokhu, liveza izici ezilandelayo: hypo- noma komzimba okukhulu, ukozela, Ukudlikizela, disorder extrapyramidal, ukushaqeka, hypotension futhi equlekile.

Okufanele ukwenze esimweni esinjalo? Kuyadingeka ukuba afeze yokwelapha ongisekelayo lingaze. Uma umuthi udle, isidingo ngokushesha iphume esiswini, kanye ukuthatha sorbent. Ngaphezu kwalokho, kubalulekile kakhulu ukusekela imisebenzi izitsha, inhliziyo futhi umgudu wokuphefumula. It is hhayi Kunconywa ukusebenzisa epinephrine njengoba kungase kuholele blood pressure ukunciphisa. izimpawu Extrapyramidal kungenzeka ukuba ayeke izidakamizwa "Biperiden" futhi nokuquleka - "Diazepam".

Ukuxhumana nezinye izidakamizwa

Lapho usebenzisa esinye isigaba ka nomuthi wathi kungase kube kukhulu imiphumela sine ka barbiturates, ethanol, nezinye izinto ezithwala okuyinto nethonya inhibitory phezu CNS.

Ukulungiselela "Flyuanksol" it is hhayi Kunconywa ukusebenzisa ngokuhlanganyela guanethidine and Drug unesimo nomphumela ofanayo. Leli qiniso kungenxa yokuthi antipsychotics kungenzeka ngempela buthaka imiphumela yabo antihypertensive.

Nge onomzali ukusetshenziswa nomuthi "Flyuanksol" kungaba ukunciphisa kusebenta izidakamizwa "levodopa" nezinye izinto ezithwala adrenergic.

Ngesikhathi esifanayo ukuthatha izidakamizwa nge "piperazine" futhi "MCP" Ngokuphawulekayo kwandisa ingozi disorder extrapyramidal.

Kufanele kuqashelwe ukuthi le izidakamizwa neuroleptic inikezwe njengoba isixazululo umjovo noma kunjalo akumelwe exutshwe olunye uketshezi.

Inani kanye analogue zomuthi

Kungakanani buyisidakamizwa "Flyuanksol"? intengo yayo impela high. Ngakho-ke, izibhebhe 50 1 mg kuzodingeka akhokhe ruble Russian mayelana 500. Uma ufuna amaphilisi 100 5 mg, bona angathengwa ruble 1,200. Njengoba for ifomu nemijovo zomuthi, kuyabiza nakakhulu. izitsha eziyisikhombisa Over 10 (20 mg / ml) kunodokotela zidinga ruble mayelana 2300.

Kuthiwani uma isiguli ayikwazi ukuthenga imithi "Flyuanksol"? analogue yayo zidayiswa cishe zonke ekhemisi ngamaketanga. Phakathi kwabo kukhona lokhu okulandelayo:

  1. Isixazululo "Flyuanksol Depot". Kuyinto ngokushesha futhi enamandla xaxa izidakamizwa. Nokho, kuyinto amaphilisi kakhulu ezibizayo.
  2. "Klopiksol" imithi. Ngo ukubaluleka liseduze kakhulu kulokho eqale iyikho. Lenza edayiswa izibhebhe futhi Izimo ambalwa.
  3. "Truksal" lisho ukuthini. Kuthengiswe amaphilisi. Inzuzo main esivuna ukusetshenziswa kwaso izingane eminyakeni-3. Izindleko kancane ngaphezu yasekuqaleni.

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